SCHEMBL10375560

SCHEMBL10375560

C=CCOc1c(C)cnc2c1CCCC2[S+]([O-])c1nc2ccccc2[nH]1

nearest known ligand 0.36

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
WDR5 P61964 1/20 0.33
KMT2A Q03164 1/20 0.33
HDAC6 Q9UBN7 1/20 0.32
KCNN3 Q9UGI6 1/20 0.32
SARM1 Q6SZW1 1/20 0.30
NPC1 O15118 1/20 0.30
RAB9A P51151 1/20 0.30
AR P10275 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10377532 0.89
SCHEMBL10376876 0.88
SCHEMBL10376878 0.88 DGAT1 (0.30)
SCHEMBL10375653 0.87 WDR5 (0.39) WDR5KMT2AHDAC6KCNN3SARM1
SCHEMBL10376875 0.87
SCHEMBL10377870 0.87 KMT2A (0.35) WDR5KMT2AHDAC6KCNN3SARM1
SCHEMBL10376797 0.86
SCHEMBL10375631 0.86 WDR5 (0.33) WDR5KMT2AHDAC6KCNN3SARM1
SCHEMBL10377506 0.83
SCHEMBL10377505 0.83

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0187977-B1 TETRAHYDROQUINOLINE DERIVATIVES, PROCESS FOR PREPARING THE SAME AND ANTI-PEPTIC ULCER COMPOSITIONS CONTAING THE SAME OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1990-08-29 EP disclosed
US-4880815-A GASTRIC JUICE INHIBITORS OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1989-11-14 US disclosed
US-4738970-A Benzimidazolyl-thio-tetrahydroquinolines and anti-peptic ulcer compositions containing the same OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1988-04-19 US disclosed
EP-0187977-A1 Tetrahydroquinoline derivatives, process for preparing the same and anti-peptic ulcer compositions containg the same OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1986-07-23 EP disclosed