SCHEMBL10375702

SCHEMBL10375702

Fc1ccc2[nH]c3c(c2c1)CN(CCCc1ccncc1)CC3

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 1/20 1.00
ACHE P22303 1/20 0.60
APAF1 O14727 1/20 0.60

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10375595 0.97 SIGMAR1 (0.94) SIGMAR1APAF1
Carvotroline SCHEMBL29710918 0.94 SIGMAR1 (0.88) SIGMAR1ACHE
Carvotroline SCHEMBL350602 0.94 SIGMAR1 (0.88) SIGMAR1ACHE
Carvotroline SCHEMBL123737 0.93 SIGMAR1 (0.86) SIGMAR1ACHE
Gevotroline SCHEMBL293396 0.88 SIGMAR1 (0.78) SIGMAR1ACHE
Gevotroline SCHEMBL30124880 0.88 SIGMAR1 (0.78) SIGMAR1ACHE
Gevotroline SCHEMBL29710901 0.88 SIGMAR1 (0.78) SIGMAR1ACHE
Gevotroline SCHEMBL120422 0.87 SIGMAR1 (0.77) SIGMAR1ACHEAPAF1
Gevotroline SCHEMBL4684544 0.87 SIGMAR1 (0.77) SIGMAR1ACHEAPAF1
Gevotroline SCHEMBL293397 0.87 SIGMAR1 (0.77) SIGMAR1ACHEAPAF1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0223344-B1 GAMMA-CARBOLINES AMERICAN HOME PRODUCTS CORPORATION (US) 1990-08-22 EP disclosed
EP-0223344-A1 Gamma-carbolines AMERICAN HOME PRODUCTS CORPORATION (US) 1987-05-27 EP disclosed