SCHEMBL10375741

SCHEMBL10375741

CC1=C(C(=O)O)C(c2csc3ncccc23)C(C(=O)O)=C(C)N1

nearest known ligand 0.38

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.38
HSD17B10 Q99714 2/20 0.38
CASP1 P29466 1/20 0.36
CACNA1B Q00975 5/20 0.36
BACE1 P56817 2/20 0.36
PDE1C Q14123 1/20 0.36
IKBKB O14920 1/20 0.35
CHUK O15111 1/20 0.35
LIMK1 P53667 1/20 0.35
IL1B P01584 1/20 0.34
MYC P01106 1/20 0.33
ALDH1A1 P00352 1/20 0.33
ADORA3 P0DMS8 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29105646 0.95 BACE1 (0.36) KDM4EHSD17B10CASP1CACNA1BBACE1
SCHEMBL30162810 0.90 BACE1 (0.38) KDM4EHSD17B10CASP1BACE1PDE1C
SCHEMBL22400637 0.90 BACE1 (0.38) KDM4EHSD17B10CASP1BACE1PDE1C
SCHEMBL22400440 0.90 ELANE (0.33) KDM4EHSD17B10BACE1IKBKBCHUK
SCHEMBL29105618 0.84 KDM4E (0.41) KDM4EHSD17B10CASP1CACNA1BPDE1C
SCHEMBL20954203 0.83 KDM4E (0.51) KDM4EHSD17B10CACNA1BPDE1CALDH1A1
SCHEMBL30489840 0.83 KDM4E (0.51) KDM4EHSD17B10CACNA1BPDE1CALDH1A1
SCHEMBL20954210 0.81 CAMKK1 (0.34) KDM4EIKBKBCHUKLIMK1ALDH1A1
SCHEMBL10372864 0.81 KDM4E (0.39) KDM4EHSD17B10CASP1CACNA1BBACE1
SCHEMBL20954247 0.79 PDE1C (0.45) KDM4EHSD17B10CASP1PDE1CALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0217530-B1 DIHYDROPYRIDINES ELI LILLY AND COMPANY (US) 1990-10-31 EP disclosed
US-4659717-A CAUSING VASODILATION ELI LILLY AND COMPANY (US) 1987-04-21 US disclosed
EP-0217530-A1 Dihydropyridines ELI LILLY AND COMPANY (US) 1987-04-08 EP disclosed