SCHEMBL10375997

SCHEMBL10375997

CC1CN(c2c(F)cc3c(=O)c(C(=O)O)cn(C4CC4)c3c2Cl)CC1NC(=O)OC(C)(C)C

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.59
POLB P06746 3/20 0.59
OPRM1 P35372 2/20 0.59
CHRM2 P08172 1/20 0.59
CHRM1 P11229 1/20 0.59
OPRD1 P41143 1/20 0.59
KDM4E B2RXH2 9/20 0.49
KCNH2 Q12809 5/20 0.49
HPGD P15428 4/20 0.49
HSD17B10 Q99714 2/20 0.49
TDP1 Q9NUW8 2/20 0.49
PRKD3 O94806 1/20 0.49
ALOX15 P16050 1/20 0.49
CLK2 P49760 1/20 0.49
CLK4 Q9HAZ1 1/20 0.49
LMNA P02545 2/20 0.47
MEN1 O00255 1/20 0.46
KMT2A Q03164 1/20 0.46
ATM Q13315 1/20 0.45
TOP2A P11388 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10681637 1.00 ALDH1A1 (0.59) ALDH1A1POLBOPRM1CHRM2CHRM1
SCHEMBL10681621 1.00 ALDH1A1 (0.59) ALDH1A1POLBOPRM1CHRM2CHRM1
SCHEMBL10687644 0.93 KCNH2 (0.51) ALDH1A1POLBOPRM1CHRM2CHRM1
SCHEMBL10374530 0.93 KCNH2 (0.51) ALDH1A1POLBOPRM1CHRM2CHRM1
SCHEMBL10687624 0.93 KCNH2 (0.51) ALDH1A1POLBOPRM1CHRM2CHRM1
SCHEMBL10375599 0.93 KCNH2 (0.51) ALDH1A1POLBOPRM1CHRM2CHRM1
SCHEMBL10375597 0.93 KCNH2 (0.51) ALDH1A1POLBOPRM1CHRM2CHRM1
SCHEMBL6215018 0.91 ALDH1A1 (0.57) ALDH1A1POLBOPRM1CHRM2CHRM1
SCHEMBL10457825 0.91 KCNH2 (0.57) ALDH1A1POLBOPRM1CHRM2CHRM1
SCHEMBL9376082 0.90 KDM4E (0.63) ALDH1A1POLBOPRM1KDM4EKCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4753953-A Pyridonecarboxylic acid derivatives and antibacterial pharmaceutical compositions thereof KYORIN PHARMACEUTICAL CO., LTD. (JP) 1988-06-28 US claimed
EP-0208210-B1 PYRIDONECARBOXYLIC ACID DERIVATIVES AND PROCESS FOR THEIR PREPARATION KYORIN PHARMACEUTICAL CO., LTD. (JP) 1990-10-24 EP disclosed
US-4753953-A Pyridonecarboxylic acid derivatives and antibacterial pharmaceutical compositions thereof KYORIN PHARMACEUTICAL CO., LTD. (JP) 1988-06-28 US disclosed
EP-0208210-A1 Pyridonecarboxylic acid derivatives and process for their preparation KYORIN PHARMACEUTICAL CO., LTD. (JP) 1987-01-14 EP disclosed