SCHEMBL10378262

SCHEMBL10378262

COC(=O)[C@@H](NC(=O)[C@@H](NC(=O)C1CCCC1)C(C)C)C(C)C

nearest known ligand 0.52

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
TSHR P16473 2/20 0.52
HPGD P15428 1/20 0.52
MAPK1 P28482 1/20 0.51
POLB P06746 1/20 0.49
CYP3A4 P08684 1/20 0.45
NPC1 O15118 1/20 0.45
ALDH1A1 P00352 1/20 0.45
TP53 P04637 1/20 0.45
MAPT P10636 1/20 0.45
RAB9A P51151 1/20 0.45
SMN1; SMN2 Q16637 2/20 0.45
PSMB5 P28074 1/20 0.43
CYP2C19 P33261 1/20 0.43
PADI1 Q9ULC6 1/20 0.41
PADI4 Q9UM07 1/20 0.41
CCR1 P32246 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27282300 1.00 TSHR (0.52) TSHRHPGDMAPK1POLBCYP3A4
Hydrochloric Acid SCHEMBL27285687 0.98 TSHR (0.51) TSHRHPGDMAPK1POLBCYP3A4
Hydrochloric Acid SCHEMBL27285688 0.98 TSHR (0.51) TSHRHPGDMAPK1POLBCYP3A4
Trifluoroacetic Acid SCHEMBL27279257 0.91 HPGD (0.46) TSHRHPGDMAPK1POLBCYP3A4
SCHEMBL7898085 0.83 TSHR (0.56) TSHRHPGDMAPK1POLBCYP3A4
SCHEMBL13525013 0.80 TSHR (0.49) TSHRPOLBALDH1A1MAPTSMN1; SMN2
SCHEMBL29789574 0.79 TSHR (0.47) TSHRHPGDMAPK1POLBALDH1A1
SCHEMBL9828504 0.79 TSHR (0.52) TSHRHPGDMAPK1POLBCYP3A4
SCHEMBL13033929 0.79 TSHR (0.47) TSHRHPGDMAPK1POLBALDH1A1
SCHEMBL9828500 0.79 TSHR (0.52) TSHRHPGDMAPK1POLBCYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1039596-A Preparation method in conjunction with the peptide of retroviral Protease SMITHKLINE BECKMAN CORP (US) 1990-02-14 CN disclosed
WO-1990000399-A1 RETROVIRAL PROTEASE BINDING PEPTIDES SMITHKLINE BECKMAN CORPORATION (US) 1990-01-25 WO disclosed