SCHEMBL10384348

SCHEMBL10384348

COc1cc(CCc2ccc(N)cc2)cc(OC)c1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 5/20 1.00
CALM1 P0DP23 4/20 0.62
AKR1B1 P15121 1/20 0.58
GFER P55789 1/20 0.56
TAAR1 Q96RJ0 1/20 0.53
TDP1 Q9NUW8 2/20 0.52
MAPK1 P28482 1/20 0.52
NQO2 P16083 1/20 0.52
TUBB4A P04350 1/20 0.50
TUBB P07437 1/20 0.50
TUBA3C P0DPH7 1/20 0.50
TUBA1B P68363 1/20 0.50
TUBA4A P68366 1/20 0.50
TUBB4B P68371 1/20 0.50
TUBB3 Q13509 1/20 0.50
TUBB2A Q13885 1/20 0.50
TUBB8 Q3ZCM7 1/20 0.50
TUBA3E Q6PEY2 1/20 0.50
TUBA1A Q71U36 1/20 0.50
TUBA1C Q9BQE3 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL9827015 0.98 CYP19A1 (0.96) CYP19A1CALM1AKR1B1GFERTAAR1
SCHEMBL8746062 0.85 CYP19A1 (0.74) CYP19A1CALM1GFERTAAR1TDP1
SCHEMBL28891744 0.85 CALM1 (0.75) CYP19A1CALM1AKR1B1TAAR1TUBB4A
SCHEMBL3364226 0.83 CYP19A1 (0.71) CYP19A1TAAR1ALDH1A1CYP3A4MAOB
SCHEMBL9491787 0.82 CYP19A1 (0.68) CYP19A1CALM1AKR1B1TAAR1TUBB4A
SCHEMBL24080182 0.80 CYP19A1 (0.67) CYP19A1GFERTDP1ALDH1A1CYP3A4
SCHEMBL4735081 0.80 CALM1 (0.73) CYP19A1CALM1AKR1B1GFERMAPK1
SCHEMBL19039706 0.80 CYP19A1 (0.67) CYP19A1CALM1TAAR1TDP1MAPK1
SCHEMBL1972535 0.79 CYP19A1 (0.66) CYP19A1CALM1AKR1B1TAAR1MAPK1
SCHEMBL153674 0.79 TAAR1 (0.64) CYP19A1CALM1AKR1B1TAAR1MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4939133-A N-substituted-2-hydroxy-α-oxo-benzeneacetamides and pharmaceutical compositions having activity as modulators of the arachidonic acid cascade WARNER-LAMBERT COMPANY (US) 1990-07-03 US disclosed