SCHEMBL1038489

SCHEMBL1038489

COCCCN1CCOc2ccc(CO[C@H]3CN(C(=O)O)C(C)[C@H](NCc4ccccc4)[C@H]3c3ccc(OC)cc3)cc21

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
THRB P10828 5/20 0.36
TP53 P04637 1/20 0.36
ALDH1A1 P00352 1/20 0.35
CYP3A4 P08684 1/20 0.35
CYP2D6 P10635 1/20 0.35
CYP2C19 P33261 1/20 0.35
MAPT P10636 4/20 0.35
REN P00797 2/20 0.34
MAOA P21397 1/20 0.34
TDP1 Q9NUW8 1/20 0.32
TSHR P16473 2/20 0.32
LMNA P02545 3/20 0.32
CACNA1G O43497 1/20 0.32
CACNA1H O95180 1/20 0.32
CACNA1I Q9P0X4 1/20 0.32
HDAC3 O15379 1/20 0.32
HDAC4 P56524 1/20 0.32
HDAC1 Q13547 1/20 0.32
HDAC7 Q8WUI4 1/20 0.32
HDAC2 Q92769 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4145756 0.88 REN (0.38) THRBTP53ALDH1A1CYP3A4CYP2D6
SCHEMBL1038928 0.84 REN (0.35) CYP3A4CYP2C19MAPTRENTDP1
SCHEMBL1038321 0.84 REN (0.34) THRBTP53MAPTRENTSHR
SCHEMBL1038354 0.83 REN (0.36) THRBALDH1A1CYP3A4CYP2D6CYP2C19
SCHEMBL1040326 0.83 REN (0.34) THRBTP53MAPTRENTSHR
SCHEMBL1040351 0.82 REN (0.35) THRBALDH1A1CYP3A4CYP2D6CYP2C19
SCHEMBL1040811 0.81 MAPT (0.33) THRBTP53ALDH1A1CYP3A4CYP2D6
SCHEMBL1039803 0.81 REN (0.34) THRBALDH1A1CYP3A4CYP2D6CYP2C19
SCHEMBL3945449 0.81 REN (0.34) THRBALDH1A1CYP3A4CYP2D6CYP2C19
SCHEMBL1038318 0.81 REN (0.37) RENMAOA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2049514-B1 NITRATE ESTERS OF PIPERIDINES NOVARTIS AG (CH) 2011-01-26 EP disclosed