SCHEMBL10399152

SCHEMBL10399152

COc1ccc(C=CC=CC(N)=O)cc1

nearest known ligand 0.63

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC8 Q9BY41 3/20 0.63
HDAC6 Q9UBN7 3/20 0.63
STAT3 P40763 1/20 0.63
F3 P13726 2/20 0.61
THRB P10828 1/20 0.59
ATM Q13315 1/20 0.59
MAOB P27338 4/20 0.58
GSK3B P49841 2/20 0.57
MAOA P21397 1/20 0.57
CYP1A2 P05177 1/20 0.57
CYP2D6 P10635 1/20 0.57
HDAC3 O15379 2/20 0.56
HDAC1 Q13547 2/20 0.56
HDAC2 Q92769 2/20 0.56
BACE1 P56817 1/20 0.53
CA1 P00915 1/20 0.52
CA2 P00918 1/20 0.52
PARP1 P09874 1/20 0.52
PARP10 Q53GL7 1/20 0.52
PARP2 Q9UGN5 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16410058 1.00 HDAC8 (0.63) HDAC8HDAC6STAT3F3THRB
SCHEMBL2009524 0.87 F3 (0.72) HDAC8HDAC6F3THRBATM
SCHEMBL1383345 0.87 F3 (0.72) HDAC8HDAC6F3THRBATM
SCHEMBL1231600 0.84 THRB (0.77) HDAC8HDAC6STAT3F3THRB
SCHEMBL2026112 0.84 HDAC8 (0.65) HDAC8HDAC6STAT3F3THRB
SCHEMBL2026113 0.84 HDAC8 (0.65) HDAC8HDAC6STAT3F3THRB
SCHEMBL1231605 0.84 THRB (0.77) HDAC8HDAC6STAT3F3THRB
SCHEMBL25307242 0.83 THRB (0.74) HDAC8HDAC6STAT3F3THRB
SCHEMBL21428246 0.83 HDAC8 (0.68) HDAC8HDAC6STAT3F3THRB
SCHEMBL13067871 0.83 HDAC8 (0.69) HDAC8HDAC6F3THRBATM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4975438-A ANTICOAGULANT HOFFMANN-LA ROCHE INC. (US) 1990-12-04 US claimed
US-4975438-A ANTICOAGULANT HOFFMANN-LA ROCHE INC. (US) 1990-12-04 US disclosed