SCHEMBL10399345

SCHEMBL10399345

CCOC(=O)c1ccc(/C=C(\C)c2ccc3c(c2)C(C)(C)CCC3(C)C)s1

nearest known ligand 0.72

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RARG P13631 15/20 0.72
RARB P10826 15/20 0.72
RARA P10276 14/20 0.72
RXRA P19793 11/20 0.72
RXRG P48443 6/20 0.72
RXRB P28702 6/20 0.72
CYP3A4 P08684 2/20 0.51
KDM4E B2RXH2 1/20 0.51
NPC1 O15118 1/20 0.51
CYP26A1 O43174 1/20 0.51
GMNN O75496 1/20 0.51
USP2 O75604 1/20 0.51
ALDH1A1 P00352 1/20 0.51
LMNA P02545 1/20 0.51
TP53 P04637 1/20 0.51
CYP1A2 P05177 1/20 0.51
POLB P06746 1/20 0.51
CYP2D6 P10635 1/20 0.51
NFKB1 P19838 1/20 0.51
CYP2C19 P33261 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10399347 1.00 RARG (0.72) RARGRARBRARARXRARXRG
SCHEMBL7219495 0.87 RXRA (0.74) RARGRARBRARARXRARXRG
SCHEMBL7219497 0.87 RXRA (0.74) RARGRARBRARARXRARXRG
SCHEMBL6428704 0.87 RARB (0.54) RARGRARBRARARXRARXRG
SCHEMBL10399193 0.83 RARB (0.51) RARGRARBRARARXRARXRG
SCHEMBL10399194 0.83 RARB (0.51) RARGRARBRARARXRARXRG
Arotinoid SCHEMBL2890175 0.81 RARG (0.70) RARGRARBRARARXRARXRG
Arotinoid SCHEMBL2890176 0.81 RARG (0.70) RARGRARBRARARXRARXRG
Arotinoid SCHEMBL29430179 0.81 RARG (0.70) RARGRARBRARARXRARXRG
SCHEMBL6427528 0.78 RXRA (0.56) RARGRARBRARARXRARXRG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4931458-A Heterocyclic rodenticidal compounds, compositions containing the compounds, and methods of use HOFFMANN-LA ROCHE INC. (US) 1990-06-05 US claimed
EP-0098591-B1 HETEROCYCLIC COMPOUNDS AND RODENTICIDES CONTAINING THEM F. HOFFMANN-LA ROCHE & CO. Aktiengesellschaft (CH) 1987-07-08 EP claimed
US-4931458-A Heterocyclic rodenticidal compounds, compositions containing the compounds, and methods of use HOFFMANN-LA ROCHE INC. (US) 1990-06-05 US disclosed
US-4816476-A BENZO(B)THIENYL GROUP OR BENZOFURAN SUBSTITUTED GROUPS HOFFMANN-LA ROCHE INC. (US) 1989-03-28 US disclosed
US-4659735-A Benzofuranyl (thienyl) propenyl derivatives useful as rodenticides HOFFMANN-LA ROCHE INC. (US) 1987-04-21 US disclosed
US-4535086-A RODENTICIDES HOFFMANN-LA ROCHE INC. (US) 1985-08-13 US disclosed