SCHEMBL7219495

SCHEMBL7219495

CCOC(=O)c1ccc(/C=C(\C)c2cc3c(cc2C)C(C)(C)CCC3(C)C)s1

nearest known ligand 0.74

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
RXRA P19793 18/20 0.74
RXRG P48443 14/20 0.74
RXRB P28702 13/20 0.74
RARB P10826 11/20 0.74
RARG P13631 9/20 0.74
RARA P10276 7/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7219497 1.00 RXRA (0.74) RXRARXRGRXRBRARBRARG
SCHEMBL10399347 0.87 RARG (0.72) RXRARXRGRXRBRARBRARG
SCHEMBL10399345 0.87 RARG (0.72) RXRARXRGRXRBRARBRARG
SCHEMBL6427528 0.87 RXRA (0.56) RXRARXRGRXRBRARBRARG
SCHEMBL3688710 0.85 RXRA (1.00) RXRARXRGRXRBRARBRARG
SCHEMBL3688709 0.85 RXRA (1.00) RXRARXRGRXRBRARBRARG
SCHEMBL3688713 0.85 RXRA (1.00) RXRARXRGRXRBRARBRARG
SCHEMBL10399194 0.83 RARB (0.51) RXRARXRGRXRBRARBRARG
SCHEMBL10399193 0.83 RARB (0.51) RXRARXRGRXRBRARBRARG
SCHEMBL7418443 0.82 RXRA (0.71) RXRARXRGRXRBRARBRARG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6624188-B1 Administered to treat or prevent one or more of the diseases and conditions selected from the group consisting of dermatoses, atherosclerosis and restenosis resulting from neointimal hyperproliferation, non-malignant and ALLERGAN, INC. 2003-09-23 US disclosed
EP-0688213-B1 TREATMENT OF TUMORS WITH COMPOUNDS HAVING RXR RETINOID RECEPTOR AGONIST ACTIVITY ALLERGAN INC (US) 2001-12-12 EP disclosed
EP-0909560-A2 Treatment o tumors with compounds having RXR retinoid receptor agoinst activity ALLERGAN, INC. (US) 1999-04-21 EP disclosed
US-5399586-A Treatment of mammals afflicted with tumors with compounds having RXR retinoid receptor agonist activity ALLERGAN, INC. (US) 1995-03-21 US disclosed
US-5324840-A Skin disorders ALLERGAN, INC. (US) 1994-06-28 US disclosed