SCHEMBL10399375

SCHEMBL10399375

O=C1C=CC(=O)C2CC=CCC12

nearest known ligand 0.37

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.37
LMNA P02545 2/20 0.37
TSHR P16473 2/20 0.37
KMT2A Q03164 2/20 0.37
HSD17B10 Q99714 2/20 0.37
TP53 P04637 2/20 0.37
CYP3A4 P08684 1/20 0.37
HPGD P15428 1/20 0.37
ALOX15 P16050 1/20 0.37
MAPK1 P28482 1/20 0.37
HTT P42858 1/20 0.37
HIF1A Q16665 1/20 0.37
NPSR1 Q6W5P4 2/20 0.35
TDP1 Q9NUW8 3/20 0.34
CA12 O43570 2/20 0.32
CA1 P00915 2/20 0.32
CA2 P00918 2/20 0.32
CA9 Q16790 2/20 0.32
POLB P06746 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11283022 1.00 ALDH1A1 (0.37) ALDH1A1LMNATSHRKMT2AHSD17B10
SCHEMBL10938530 0.69 MAPT (0.33) ALDH1A1KMT2AHPGD
SCHEMBL7123770 0.69 ALDH1A1 (0.37) ALDH1A1LMNATSHRKMT2AHSD17B10
SCHEMBL1628615 0.69 ALDH1A1 (0.37) ALDH1A1LMNATSHRKMT2AHSD17B10
SCHEMBL10937868 0.68 MAPT (0.33) ALDH1A1KMT2AHPGD
SCHEMBL10935590 0.68 MAPT (0.33) ALDH1A1KMT2AHPGD
SCHEMBL4560700 0.67
SCHEMBL9632348 0.67 PDE4A (0.38) ALDH1A1LMNATSHRKMT2AHSD17B10
SCHEMBL5160089 0.67 ALDH1A1 (0.35) ALDH1A1LMNATSHRKMT2AHSD17B10
SCHEMBL4475890 0.67 NLRP3 (0.33)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 15 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0007403-B1 5,12-DIHYDROXY-1,2,3,4,6,11-HEXAHYDRO-2,6,11-TRIOXONAPHTHACENES AND THEIR SYNTHESIS THE UNIVERSITY OF KANSAS (US) 1982-11-24 EP claimed
US-4244880-A Anthracycline synthesis UNIVERSITY OF KANSAS ENDOWMENT ASSOCIATION (US) 1981-01-13 US claimed
EP-0007403-A1 5,12-dihydroxy-1,2,3,4,6,11-hexahydro-2,6,11-trioxonaphthacenes and their synthesis THE UNIVERSITY OF KANSAS (US) 1980-02-06 EP claimed
WO-2015089349-A1 INHIBITION OF ISOPRENOID BIOSYNTHETIC PATHWAYS TO TREAT NEUROINFLAMMATORY DISORDERS TABACZYNSKI DAVID A (US) 2015-06-18 WO disclosed
CN-101885674-B Preparation method of 5,8-dimethoxy-2-tetralin ketone GANSU HAOTIAN CHEMEXPRESS CO LTD 2015-03-11 CN disclosed
CN-101885674-A Preparation method of 5,8-dimethoxy-2-tetralin ketone GANSU HAOTIAN CHEMEXPRESS CO LTD 2010-11-17 CN disclosed
US-4975461-A Enzymes/oxidoreductases/inhibitors E. R. SQUIBB & SONS, INC. (US) 1990-12-04 US disclosed
EP-0136893-B1 Benzo[a]phenothiazines and hydro-derivatives and pharmaceutical compositions containing them MERCK FROSST CANADA INC. (CA) 1989-08-16 EP disclosed
EP-0007403-B1 5,12-DIHYDROXY-1,2,3,4,6,11-HEXAHYDRO-2,6,11-TRIOXONAPHTHACENES AND THEIR SYNTHESIS THE UNIVERSITY OF KANSAS (US) 1982-11-24 EP disclosed
EP-0043435-A1 Intermediate products occurring in anthracycline synthesis THE UNIVERSITY OF KANSAS (US) 1982-01-13 EP disclosed
US-4267373-A HYDROXY- OR -OXY-SUBSTITUTED-6-ALKYL- OR DIALKYLAMINO-7-HYDROXY DERIVATIVES E. R. SQUIBB & SONS, INC. (US) 1981-05-12 US disclosed
US-4244880-A Anthracycline synthesis UNIVERSITY OF KANSAS ENDOWMENT ASSOCIATION (US) 1981-01-13 US disclosed
EP-0007404-A1 Synthesis of 2-hydroxy-2-acetyl-1,2,3,4-tetrahydronaphthalene compounds THE UNIVERSITY OF KANSAS (US) 1980-02-06 EP disclosed
EP-0007403-A1 5,12-dihydroxy-1,2,3,4,6,11-hexahydro-2,6,11-trioxonaphthacenes and their synthesis THE UNIVERSITY OF KANSAS (US) 1980-02-06 EP disclosed
US-4076843-A 5,6,7,8-Tetrahydronaphthalene hypotensive agents E. R. SQUIBB & SONS, INC. (US) 1978-02-28 US disclosed