SCHEMBL10399462

SCHEMBL10399462

COc1ccc2c(c1)CCC(Nc1ccc(O)cc1)C2

nearest known ligand 0.58

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CYP26A1 O43174 2/20 0.58
CA1 P00915 6/20 0.57
CA2 P00918 6/20 0.57
ACHE P22303 6/20 0.57
MTNR1A P48039 1/20 0.54
MTNR1B P49286 1/20 0.54
DRD2 P14416 4/20 0.51
DRD3 P35462 4/20 0.51
CYP24A1 Q07973 1/20 0.44
GRIN1 Q05586 1/20 0.44
GRIN2B Q13224 1/20 0.44
CYP19A1 P11511 1/20 0.43
HDAC8 Q9BY41 1/20 0.42
KCNH2 Q12809 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10398545 0.89 CYP26A1 (0.50) CYP26A1CA1CA2ACHEMTNR1A
SCHEMBL11851549 0.86 CA1 (0.57) CYP26A1CA1CA2ACHEMTNR1A
SCHEMBL10398507 0.84 CA1 (0.56) CA1CA2ACHEDRD2DRD3
SCHEMBL10398569 0.84 HDAC8 (0.43) CYP26A1CA1CA2ACHEMTNR1A
SCHEMBL10399481 0.82 GRIN1 (0.54) CYP26A1CA1CA2ACHEDRD2
SCHEMBL8624827 0.79 CA1 (0.64) CYP26A1CA1CA2ACHEMTNR1A
SCHEMBL8237115 0.79 CA1 (0.64) CYP26A1CA1CA2ACHEMTNR1A
SCHEMBL8624829 0.79 CA1 (0.64) CYP26A1CA1CA2ACHEMTNR1A
Hydrochloric Acid SCHEMBL10851134 0.77 CA1 (0.63) CYP26A1CA1CA2ACHEMTNR1A
SCHEMBL10399460 0.77 MTNR1A (0.51) CA1CA2MTNR1AMTNR1BDRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4975461-A Enzymes/oxidoreductases/inhibitors E. R. SQUIBB & SONS, INC. (US) 1990-12-04 US disclosed