SCHEMBL10399481

SCHEMBL10399481

COc1ccc2c(c1)CCC(Nc1ccc(OCc3ccccc3)cc1)C2

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRIN1 Q05586 1/20 0.54
GRIN2B Q13224 1/20 0.54
KDM1A O60341 1/20 0.51
MAOA P21397 1/20 0.51
MAOB P27338 1/20 0.51
CA1 P00915 2/20 0.48
CA2 P00918 2/20 0.48
ACHE P22303 2/20 0.48
SIGMAR1 Q99720 1/20 0.47
DRD2 P14416 2/20 0.47
DRD3 P35462 2/20 0.47
HRH3 Q9Y5N1 2/20 0.47
FAAH O00519 4/20 0.47
TAOK1 Q7L7X3 1/20 0.47
TAOK3 Q9H2K8 1/20 0.47
SMN1; SMN2 Q16637 2/20 0.47
ALDH1A1 P00352 1/20 0.47
GAA P10253 1/20 0.47
MAPT P10636 1/20 0.47
ALOX12 P18054 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10399771 0.91 AR (0.50) GRIN1GRIN2BKDM1AMAOAMAOB
SCHEMBL10400090 0.89 KDM1A (0.52) GRIN1GRIN2BKDM1AMAOAMAOB
SCHEMBL10399768 0.87 TAOK1 (0.55) GRIN2BSIGMAR1HRH3TAOK1TAOK3
SCHEMBL11851549 0.87 CA1 (0.57) GRIN1GRIN2BCA1CA2ACHE
SCHEMBL10399462 0.82 CYP26A1 (0.58) GRIN1GRIN2BCA1CA2ACHE
SCHEMBL10399740 0.81 ALDH1A1 (0.47) KDM1AMAOAMAOBCA1CA2
SCHEMBL10398571 0.80 CYP1A2 (0.50) MAOAMAOBTAOK1TAOK3SMN1; SMN2
SCHEMBL12524812 0.79 GRIN2B (0.66) GRIN1GRIN2BCA1CA2ACHE
SCHEMBL12614692 0.76 LTA4H (0.55) KDM1AMAOAMAOBSMN1; SMN2GAA
Hydrochloric Acid SCHEMBL27903791 0.75 LTA4H (0.54) KDM1AMAOAMAOBSMN1; SMN2GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4975461-A Enzymes/oxidoreductases/inhibitors E. R. SQUIBB & SONS, INC. (US) 1990-12-04 US disclosed