SCHEMBL10399962

SCHEMBL10399962

COc1ccc(-n2ccc3ccccc32)cc1Cl

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BIRC5 O15392 1/20 0.55
MAPT P10636 4/20 0.51
ALDH1A1 P00352 2/20 0.51
RAB9A P51151 2/20 0.51
ALOX15 P16050 1/20 0.51
SMN1; SMN2 Q16637 1/20 0.51
HSD17B10 Q99714 1/20 0.51
EGFR P00533 1/20 0.43
TUBB4A P04350 1/20 0.43
TUBB P07437 1/20 0.43
TUBA3C P0DPH7 1/20 0.43
TUBA1B P68363 1/20 0.43
TUBA4A P68366 1/20 0.43
TUBB4B P68371 1/20 0.43
TUBB3 Q13509 1/20 0.43
TUBB2A Q13885 1/20 0.43
TUBB8 Q3ZCM7 1/20 0.43
TUBA3E Q6PEY2 1/20 0.43
TUBA1A Q71U36 1/20 0.43
TUBA1C Q9BQE3 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10400222 0.82 BIRC5 (0.47) BIRC5ALDH1A1RAB9ASMN1; SMN2EGFR
SCHEMBL28780185 0.82 BIRC5 (0.47) BIRC5MAPTALDH1A1RAB9ASMN1; SMN2
SCHEMBL16296617 0.79 BIRC5 (0.47) BIRC5MAPTTUBB4ATUBBTUBA3C
SCHEMBL20604726 0.79 FFAR4 (0.44) MAPTALDH1A1RAB9AALOX15SMN1; SMN2
SCHEMBL5662515 0.75 FGFR1 (0.55) BIRC5MAPTALDH1A1RAB9ASMN1; SMN2
SCHEMBL1078090 0.74 BIRC5 (0.61) BIRC5MAPTALDH1A1RAB9ASMN1; SMN2
SCHEMBL29896757 0.74 BIRC5 (0.61) BIRC5MAPTALDH1A1RAB9ASMN1; SMN2
SCHEMBL16296928 0.74 BIRC5 (0.40) BIRC5EGFRTUBB4ATUBBTUBA3C
SCHEMBL20201236 0.73 ALDH1A1 (0.57) MAPTALDH1A1RAB9AALOX15SMN1; SMN2
SCHEMBL6190919 0.72 BIRC5 (0.61) BIRC5MAPTALDH1A1CYP19A1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4977178-A Method of treating anxiety and depression with 1-phenyl-2(1H,3H)-indolone psycho-therapeutic agents PFIZER INC. (US) 1990-12-11 US disclosed
US-4879391-A 1-Phenyl-2(1H,3H)-indolone psychotherapeutic agents PFIZER INC. (US) 1989-11-07 US disclosed
US-4861880-A 1-phenyl-2(1H,3H)-indolone psycho-therapeutic agents PFIZER INC. (US) 1989-08-29 US disclosed
EP-0104860-B1 1-PHENYL-2(1H,3H)-INDOLONE PSYCHO-THERAPEUTIC AGENTS PFIZER INC. (US) 1987-03-18 EP disclosed
US-4476307-A Heteroylidene indolone compounds PFIZER INC. (US) 1984-10-09 US disclosed
EP-0104860-A1 1-Phenyl-2(1H,3H)-indolone psycho-therapeutic agents PFIZER INC. (US) 1984-04-04 EP disclosed