SCHEMBL10401660

SCHEMBL10401660

CCOC(=O)C(=O)Nc1ccc(C=Cc2ccc3ccccc3n2)cc1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRM4 Q14833 1/20 0.57
CYSLTR2 Q9NS75 3/20 0.52
CYSLTR1 Q9Y271 3/20 0.52
MAPT P10636 7/20 0.51
RAB9A P51151 5/20 0.51
KDM4E B2RXH2 4/20 0.51
NPC1 O15118 4/20 0.51
SMN1; SMN2 Q16637 4/20 0.51
LMNA P02545 3/20 0.51
L3MBTL1 Q9Y468 3/20 0.51
MEN1 O00255 2/20 0.51
KMT2A Q03164 2/20 0.51
ALDH1A1 P00352 2/20 0.51
PKM P14618 1/20 0.49
MAPK1 P28482 2/20 0.48
RXFP1 Q9HBX9 1/20 0.48
CYP19A1 P11511 2/20 0.46
HTT P42858 2/20 0.46
HDAC3 O15379 1/20 0.46
HDAC4 P56524 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10401659 1.00 GRM4 (0.57) GRM4CYSLTR2CYSLTR1MAPTRAB9A
SCHEMBL28435833 0.82 RAB9A (0.65) CYSLTR2CYSLTR1MAPTRAB9AKDM4E
SCHEMBL28435835 0.82 RAB9A (0.65) CYSLTR2CYSLTR1MAPTRAB9AKDM4E
SCHEMBL1246543 0.78 KDM4E (0.57) CYSLTR2CYSLTR1MAPTRAB9AKDM4E
SCHEMBL1244748 0.77 KDM4E (0.56) CYSLTR2CYSLTR1MAPTRAB9AKDM4E
SCHEMBL1246644 0.76 MAPT (0.54) CYSLTR2CYSLTR1MAPTRAB9AKDM4E
SCHEMBL10444695 0.76 NPC1 (0.55) RAB9AKDM4ENPC1SMN1; SMN2MEN1
Hydrochloric Acid SCHEMBL9779738 0.74 HPGD (0.53) GRM4MAPTRAB9AKDM4ENPC1
SCHEMBL20921524 0.74 RAB9A (0.68) CYSLTR2CYSLTR1MAPTRAB9AKDM4E
SCHEMBL6483597 0.74 RAB9A (0.68) CYSLTR2CYSLTR1MAPTRAB9AKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4962203-A ANTIASTHMATIC, ANTIALLERGENIC, ANTIINFLAMMATORY AND CYTOPROTECTIVE AGENTS MERCK FROST CANADA, INC. (CA) 1990-10-09 US disclosed
EP-0206751-A2 2-Substituted quinolines, their preparation and use MERCK FROSST CANADA INC. (CA) 1986-12-30 EP disclosed