SCHEMBL10406376

SCHEMBL10406376

C=CC[C@H]1C=CC(=O)C[C@@H]1C

nearest known ligand 0.33

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
NOS3 P29474 1/20 0.33
NOS2 P35228 1/20 0.33
NFKB1 P19838 3/20 0.32
NFKB2 Q00653 3/20 0.32
RELA Q04206 3/20 0.32
L3MBTL1 Q9Y468 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10406379 1.00 NOS3 (0.33) NOS3NOS2NFKB1NFKB2RELA
SCHEMBL10406377 1.00 NOS3 (0.33) NOS3NOS2NFKB1NFKB2RELA
SCHEMBL10406774 0.83
SCHEMBL10406776 0.83
SCHEMBL11058198 0.79 NFKB1 (0.33) NFKB1NFKB2RELA
SCHEMBL15418719 0.77 NFKB1 (0.38) NFKB1NFKB2RELA
SCHEMBL15480919 0.73
SCHEMBL11237892 0.71 NFKB1 (0.33) NFKB1NFKB2RELA
SCHEMBL13766089 0.68
SCHEMBL11060621 0.67 NOS3 (0.35) NOS3NOS2L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4921994-A ANALGESICS, ANTIEMETICS PFIZER INC. (US) 1990-05-01 US disclosed
US-4831059-A ANTIEMETICS; DIARRHEA; CENTRAL NERVOUS SYSTEM PFIZER INC. (US) 1989-05-16 US disclosed
EP-0048572-B1 SUBSTITUTED 2-HYDROXYPHENYL CYCLOALKANES AND PHARMACEUTICAL COMPOSITIONS THEREOF PFIZER INC. (US) 1987-07-15 EP disclosed
US-4371720-A ANTIDIARRHEALS, ANTIEMETICS PFIZER INC. (US) 1983-02-01 US disclosed