SCHEMBL10415151

SCHEMBL10415151

FC(F)(F)C(F)(F)C(F)(F)/C=C/c1ccccc1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAOB P27338 3/20 0.42
NFE2L2 Q16236 5/20 0.41
CYP2C19 P33261 1/20 0.40
GRM4 Q14833 1/20 0.38
ALDH1A1 P00352 4/20 0.37
TSHR P16473 1/20 0.37
LMNA P02545 3/20 0.37
TRPA1 O75762 2/20 0.37
CYP19A1 P11511 1/20 0.37
MAOA P21397 1/20 0.37
ALOX5 P09917 1/20 0.37
MAPK1 P28482 1/20 0.37
MAPT P10636 2/20 0.37
S1PR4 O95977 1/20 0.37
S1PR1 P21453 1/20 0.37
NPSR1 Q6W5P4 1/20 0.37
CYP1A1 P04798 1/20 0.36
CYP1B1 Q16678 1/20 0.36
HDAC3 O15379 1/20 0.35
TNKS O95271 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10415153 1.00 MAOB (0.42) MAOBNFE2L2CYP2C19GRM4ALDH1A1
SCHEMBL5352063 0.94 MAOB (0.41) MAOBNFE2L2CYP2C19GRM4ALDH1A1
SCHEMBL10522046 0.94 MAOB (0.41) MAOBNFE2L2CYP2C19GRM4ALDH1A1
SCHEMBL9222592 0.92 MAOB (0.39) MAOBNFE2L2CYP2C19GRM4ALDH1A1
SCHEMBL16439911 0.86 MAOB (0.46) MAOBNFE2L2CYP2C19GRM4ALDH1A1
SCHEMBL16439910 0.86 MAOB (0.46) MAOBNFE2L2CYP2C19GRM4ALDH1A1
SCHEMBL6862118 0.83 CYP2C19 (0.42) MAOBNFE2L2CYP2C19GRM4ALDH1A1
SCHEMBL7174980 0.81 ALDH1A1 (0.43) MAOBNFE2L2CYP2C19ALDH1A1TSHR
SCHEMBL7868570 0.80 NPC1 (0.40) NFE2L2CYP2C19ALDH1A1LMNAMAPT
SCHEMBL3854993 0.78 ALDH1A1 (0.48) MAOBNFE2L2CYP2C19GRM4ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4956123-A REACTING A STYRENE TYPE COMPOUND WITH A DIHALOACYL PEROXIDE TO MAKE A FLUOROALKYLAROMATIC ESTER NIPPON OILS & FATS COMPANY, LTD. (JP) 1990-09-11 US disclosed
EP-0189275-B1 METHOD FOR MANUFACTURE OF FLUORINE-CONTAINING AROMATIC DERIVATIVES NIPPON OIL AND FATS COMPANY, LIMITED (JP) 1989-10-18 EP disclosed
EP-0189275-A2 Method for manufacture of fluorine-containing aromatic derivatives NIPPON OIL AND FATS COMPANY, LIMITED (JP) 1986-07-30 EP disclosed