SCHEMBL10429048

SCHEMBL10429048

Nc1cnccc1NCc1ccc(F)cc1

nearest known ligand 0.54

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.54
KDM4E B2RXH2 2/20 0.54
HPGD P15428 1/20 0.54
KCNH3 Q9ULD8 3/20 0.47
GPR55 Q9Y2T6 1/20 0.46
L3MBTL1 Q9Y468 1/20 0.42
BRD4 O60885 1/20 0.42
KAT2B Q92831 1/20 0.42
RPS6KB1 P23443 1/20 0.41
HTT P42858 1/20 0.41
APP P05067 1/20 0.40
POLB P06746 1/20 0.40
KDM4C Q9H3R0 2/20 0.40
KDM6B O15054 1/20 0.40
KDM4A O75164 1/20 0.40
KDM4D Q6B0I6 1/20 0.40
KDM5B Q9UGL1 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11098575 0.87 ALDH1A1 (0.54) ALDH1A1KDM4EHPGDKCNH3GPR55
Hydrochloric Acid SCHEMBL10508061 0.86 ALDH1A1 (0.53) ALDH1A1KDM4EHPGDKCNH3GPR55
SCHEMBL8249024 0.84 CA12 (0.49) ALDH1A1KDM4EHPGDRPS6KB1KDM4C
SCHEMBL16489567 0.84 KDM4E (0.54) ALDH1A1KDM4EHPGDRPS6KB1APP
SCHEMBL16489564 0.83 KDM4C (0.56) ALDH1A1KDM4EHPGDKCNH3HTT
SCHEMBL4718906 0.83 ASPH (0.45) KDM4EAPP
SCHEMBL16489574 0.83 MEN1 (0.47) ALDH1A1KDM4EHPGDRPS6KB1
SCHEMBL7012861 0.79 RPS6KB1 (0.55) ALDH1A1KDM4EHPGDL3MBTL1RPS6KB1
SCHEMBL9134263 0.76 HDAC1 (0.49) ALDH1A1KDM4EKCNH3APP
SCHEMBL16489576 0.75 MAP4K4 (0.47) ALDH1A1KDM4EHPGDKCNH3L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0151824-B1 N-(4-PIPERIDINYL) BICYCLIC CONDENSED 2-IMIDAZOLAMINE DERIVATIVES JANSSEN PHARMACEUTICA N.V. (BE) 1990-04-04 EP disclosed
EP-0099139-B1 NOVEL N-(BICYCLIC HETEROCYCLYL)-4-PIPERIDINAMINES JANSSEN PHARMACEUTICA N.V. (BE) 1987-02-11 EP disclosed
EP-0151824-A2 N-(4-piperidinyl) bicyclic condensed 2-imidazolamine derivatives JANSSEN PHARMACEUTICA N.V. (BE) 1985-08-21 EP disclosed
EP-0151826-A1 4-[(Bicyclic heterocyclyl)-methyl and -hetero]-piperidines JANSSEN PHARMACEUTICA N.V. (BE) 1985-08-21 EP disclosed