SCHEMBL10429321

SCHEMBL10429321

Cc1cccc(-c2nsc3c(=O)[nH]nnc23)c1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA3 P0DMS8 1/20 0.39
NOTUM Q6P988 1/20 0.39
NPC1 O15118 3/20 0.36
RAB9A P51151 3/20 0.36
ALDH1A1 P00352 2/20 0.36
SMN1; SMN2 Q16637 2/20 0.36
MAPT P10636 1/20 0.36
NFKB1 P19838 1/20 0.36
NFKB2 Q00653 1/20 0.36
RELA Q04206 1/20 0.36
HTR7 P34969 1/20 0.35
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35
XDH P47989 1/20 0.35
MAPK14 Q16539 3/20 0.34
CYP1A2 P05177 1/20 0.34
CYP2C9 P11712 1/20 0.34
PBRM1 Q86U86 1/20 0.34
GRIN2D O15399 1/20 0.34
GRIN3B O60391 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10429364 0.86 NOTUM (0.33) NOTUMALDH1A1MEN1KMT2AHPGD
SCHEMBL10429331 0.85 NOTUM (0.43) NOTUMALDH1A1SMN1; SMN2MEN1KMT2A
SCHEMBL10429361 0.84 MAOB (0.36) NPC1RAB9AALDH1A1SMN1; SMN2MAPT
SCHEMBL10429298 0.84 NOTUM (0.39) ADORA3NOTUMHTR7GRIN2DGRIN3B
SCHEMBL10429312 0.84 NOTUM (0.39) ADORA3NOTUMHTR7
SCHEMBL10429305 0.84 NOTUM (0.42) NOTUMALDH1A1SMN1; SMN2MAPTMEN1
SCHEMBL2121780 0.83 NPSR1 (0.40) NPC1RAB9AALDH1A1SMN1; SMN2MEN1
SCHEMBL7166444 0.81 NOTUM (0.42) NOTUMRAB9AALDH1A1SMN1; SMN2XDH
SCHEMBL10429323 0.81 MAOB (0.40) NOTUMXDH
SCHEMBL17968384 0.79 TSHR (0.46) ADORA3NPC1RAB9AALDH1A1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4920119-A XANTHINE OXIDASE INHIBITORS; CONTROL OR PREVENTION OF GOUT OR ISCHEMIA HOFFMANN-LA ROCHE INC. (US) 1990-04-24 US disclosed
EP-0274654-A2 1,2,3-Triazin-4(3H)-one derivatives, process for their preparation and medicaments containing them F. HOFFMANN-LA ROCHE AG (CH) 1988-07-20 EP disclosed