SCHEMBL10429323

SCHEMBL10429323

N#Cc1cccc(-c2nsc3c(=O)[nH]nnc23)c1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAOB P27338 2/20 0.40
XDH P47989 1/20 0.38
PGR P06401 4/20 0.38
CLK4 Q9HAZ1 1/20 0.38
ADORA2A P29274 3/20 0.37
ADORA1 P30542 2/20 0.37
IDO1 P14902 2/20 0.36
NOTUM Q6P988 1/20 0.36
MAP4K4 O95819 1/20 0.36
GSK3A P49840 1/20 0.36
KDM5B Q9UGL1 1/20 0.36
TDO2 P48775 1/20 0.36
GABRA1 P14867 1/20 0.35
GABRG2 P18507 1/20 0.35
GABRB3 P28472 1/20 0.35
GABRA5 P31644 1/20 0.35
GABRA3 P34903 1/20 0.35
ADORA2B P29275 1/20 0.35
CHEK1 O14757 1/20 0.35
CFTR P13569 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10429312 0.81 NOTUM (0.39) MAOBADORA2AADORA1IDO1NOTUM
SCHEMBL10429321 0.81 ADORA3 (0.39) XDHNOTUM
SCHEMBL10429361 0.81 MAOB (0.36) MAOBIDO1
SCHEMBL10429298 0.81 NOTUM (0.39) MAOBPGRADORA2AADORA1IDO1
SCHEMBL2121780 0.80 NPSR1 (0.40) XDHIDO1
SCHEMBL10429331 0.79 NOTUM (0.43) IDO1NOTUM
SCHEMBL10429305 0.78 NOTUM (0.42) MAOBXDHPGRNOTUM
SCHEMBL7166444 0.78 NOTUM (0.42) MAOBXDHADORA2AADORA1IDO1
SCHEMBL10429340 0.76 NOTUM (0.39) MAOBADORA2AADORA1NOTUM
SCHEMBL10429356 0.76 ALDH1A1 (0.32) XDH

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0274654-A2 1,2,3-Triazin-4(3H)-one derivatives, process for their preparation and medicaments containing them F. HOFFMANN-LA ROCHE AG (CH) 1988-07-20 EP claimed
US-4920119-A XANTHINE OXIDASE INHIBITORS; CONTROL OR PREVENTION OF GOUT OR ISCHEMIA HOFFMANN-LA ROCHE INC. (US) 1990-04-24 US disclosed
EP-0274654-A2 1,2,3-Triazin-4(3H)-one derivatives, process for their preparation and medicaments containing them F. HOFFMANN-LA ROCHE AG (CH) 1988-07-20 EP disclosed