SCHEMBL1043069

SCHEMBL1043069

C[C@@H]1COc2ccc(F)cc2O1

nearest known ligand 0.45

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
LTA4H P09960 2/20 0.45
CA2 P00918 1/20 0.41
DRD2 P14416 1/20 0.41
AKR1B1 P15121 3/20 0.40
CYP19A1 P11511 1/20 0.39
FFAR1 O14842 1/20 0.37
HCRTR2 O43614 1/20 0.36
DAO P14920 1/20 0.36
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35
ALOX5 P09917 3/20 0.35
NR3C1 P04150 1/20 0.34
PGR P06401 1/20 0.34
NR3C2 P08235 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19393060 1.00 LTA4H (0.45) LTA4HCA2DRD2AKR1B1CYP19A1
SCHEMBL1042716 1.00 LTA4H (0.45) LTA4HCA2DRD2AKR1B1CYP19A1
SCHEMBL8344689 0.79 CA2 (0.49) CA2AKR1B1CYP19A1FFAR1MEN1
SCHEMBL1043313 0.79 AKR1B1 (0.40) LTA4HAKR1B1
SCHEMBL1043068 0.78 LTA4H (0.45) LTA4HCA2DRD2AKR1B1CYP19A1
SCHEMBL30438928 0.78 CHRNB4 (0.52) DRD2
SCHEMBL16656033 0.78 PBRM1 (0.50) CA2AKR1B1CYP19A1FFAR1HCRTR2
SCHEMBL1044542 0.78 PBRM1 (0.50) CA2AKR1B1CYP19A1FFAR1HCRTR2
SCHEMBL1877576 0.78 CA2 (0.48) CA2DRD2AKR1B1CYP19A1FFAR1
SCHEMBL1879365 0.78 CHRNB4 (0.52) DRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2271635-A1 MODULATORS OF DOPAMINE NEUROTRANSMISSION NSAB, Filial af NeuroSearch Sweden AB, Sverige (DK) 2011-01-12 EP disclosed
WO-2009133109-A1 MODULATORS OF DOPAMINE NEUROTRANSMISSION NSAB, FILIAL AF NEUROSEARCH SWEDEN AB, SVERIGE (DK) 2009-11-05 WO disclosed