SCHEMBL10436624

SCHEMBL10436624

FC(F)(F)c1ccc2ncccc2c1.O=[N+]([O-])c1cc2ccc1-2

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TRPV1 Q8NER1 1/20 0.45
NFKBIA P25963 1/20 0.45
RELA Q04206 1/20 0.45
SLC40A1 Q9NP59 1/20 0.45
NPC1 O15118 1/20 0.43
POLB P06746 1/20 0.43
RAB9A P51151 1/20 0.43
MAPT P10636 4/20 0.42
ALDH1A1 P00352 3/20 0.42
LMNA P02545 1/20 0.42
GAA P10253 1/20 0.42
HPGD P15428 1/20 0.42
L3MBTL1 Q9Y468 1/20 0.41
TOP1 P11387 2/20 0.41
MET P08581 2/20 0.40
KDM4E B2RXH2 1/20 0.40
TRPM8 Q7Z2W7 1/20 0.39
AKR1C3 P42330 1/20 0.39
AKR1C2 P52895 1/20 0.39
PTGES O14684 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1538451 0.79 NPC1 (0.57) NPC1POLBRAB9AMAPTALDH1A1
SCHEMBL30038760 0.79 NPC1 (0.57) NPC1POLBRAB9AMAPTALDH1A1
SCHEMBL10436779 0.79 NPC1 (0.49) TRPV1SLC40A1NPC1POLBRAB9A
SCHEMBL2976577 0.74 CYP11B1 (0.48) NPC1MAPTALDH1A1LMNAKDM4E
SCHEMBL30340906 0.73 NPC1 (0.70) TRPV1NPC1POLBRAB9AMAPT
SCHEMBL2963618 0.72 ALDH1A1 (0.56) NPC1POLBRAB9AMAPTALDH1A1
SCHEMBL5445828 0.71 HSP90AA1 (0.62) NFKBIARELASLC40A1NPC1POLB
SCHEMBL14539004 0.71 NPC1 (0.66) NPC1POLBRAB9AMAPTALDH1A1
Quinoline SCHEMBL17439118 0.70 ALDH1A1 (0.49) NPC1POLBRAB9AMAPTALDH1A1
SCHEMBL31511355 0.69 ALDH1A1 (0.50) NPC1POLBRAB9AMAPTALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0354994-A2 Quinoline derivatives, their production and use Takeda Chemical Industries, Ltd. (JP) 1990-02-21 EP disclosed