SCHEMBL1044092

SCHEMBL1044092

CC(=O)SC1CCCC1(CCCNC(=O)OCc1ccccc1)C(=O)O

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KEAP1 Q14145 3/20 0.48
NFE2L2 Q16236 3/20 0.48
HTT P42858 1/20 0.46
MEN1 O00255 1/20 0.44
KMT2A Q03164 1/20 0.44
LMNA P02545 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
TGM2 P21980 1/20 0.43
ALDH1A1 P00352 1/20 0.41
L3MBTL1 Q9Y468 2/20 0.40
DPP8 Q6V1X1 2/20 0.40
DPP7 Q9UHL4 2/20 0.40
DPP4 P27487 1/20 0.40
DPP9 Q86TI2 1/20 0.40
MAPT P10636 1/20 0.39
IDO1 P14902 1/20 0.39
TDO2 P48775 1/20 0.39
CTSL P07711 1/20 0.38
CTSB P07858 1/20 0.38
CTSS P25774 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3784529 1.00 KEAP1 (0.48) KEAP1NFE2L2HTTMEN1KMT2A
SCHEMBL3790848 0.93 KEAP1 (0.47) KEAP1NFE2L2HTTMEN1KMT2A
SCHEMBL3778653 0.93 KEAP1 (0.47) KEAP1NFE2L2HTTMEN1KMT2A
SCHEMBL3788955 0.93 KEAP1 (0.47) KEAP1NFE2L2HTTMEN1KMT2A
SCHEMBL1041146 0.83 HTT (0.51) KEAP1NFE2L2HTTMEN1KMT2A
SCHEMBL1077185 0.80 HTT (0.46) KEAP1NFE2L2HTTMEN1KMT2A
SCHEMBL3787513 0.78 HTT (0.50) KEAP1NFE2L2HTTMEN1KMT2A
SCHEMBL3787712 0.75 HTT (0.45) KEAP1NFE2L2HTTMEN1KMT2A
SCHEMBL3790851 0.72 HTT (0.46) KEAP1NFE2L2HTTMEN1KMT2A
SCHEMBL3778657 0.72 HTT (0.46) KEAP1NFE2L2HTTMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2272826-A1 2-mercaptopentancarboxylic acid derivatives, the method for preparing them and the pharmaceutical compositions containing them Les Laboratoires Servier (FR) 2011-01-12 EP disclosed
WO-2010149888-A1 DERIVATIVES OF 2-MERCAPTOCYCLOPENTANE CARBOXYLIC ACID, METHOD FOR THE PREPARATION THEREOF, AND PHARMACEUTICAL COMPOSITIONS CONTAINING THE SAME LES LABORATOIRES SERVIER (FR) 2010-12-29 WO disclosed