SCHEMBL10445864

SCHEMBL10445864

O=C(O)c1cn(-c2ccc(F)cc2)c2ccccc2c1=O

nearest known ligand 0.66

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
LMNA P02545 4/20 0.66
KDM4E B2RXH2 4/20 0.66
MEN1 O00255 2/20 0.54
KMT2A Q03164 2/20 0.54
ALDH1A1 P00352 2/20 0.54
RORC P51449 6/20 0.53
HPGD P15428 1/20 0.53
HSD17B10 Q99714 1/20 0.53
TP53 P04637 1/20 0.50
NR4A2 P43354 1/20 0.49
HDAC1 Q13547 1/20 0.48
HDAC2 Q92769 1/20 0.48
CYP1A2 P05177 1/20 0.48
CYP2C9 P11712 1/20 0.48
CHRM1 P11229 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30309505 1.00 LMNA (0.66) LMNAKDM4EMEN1KMT2AALDH1A1
SCHEMBL2610312 0.90 KDM4E (0.71) LMNAKDM4EMEN1KMT2AALDH1A1
SCHEMBL5100563 0.90 KDM4E (0.61) LMNAKDM4ERORCNR4A2CYP1A2
SCHEMBL30309433 0.90 KDM4E (0.61) LMNAKDM4ERORCNR4A2CYP1A2
SCHEMBL16207451 0.87 LMNA (0.53) LMNAKDM4EMEN1KMT2AALDH1A1
SCHEMBL17883637 0.87 LMNA (0.53) LMNAKDM4EMEN1KMT2AALDH1A1
SCHEMBL30309442 0.87 LMNA (0.53) LMNAKDM4EMEN1KMT2AALDH1A1
SCHEMBL4079943 0.86 LMNA (0.55) LMNAKDM4ERORCNR4A2CYP1A2
SCHEMBL10516924 0.86 LMNA (0.60) LMNAKDM4EMEN1KMT2AALDH1A1
SCHEMBL30309390 0.86 LMNA (0.55) LMNAKDM4ERORCNR4A2CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115784987-A Compound related to pneumonia, preparation method and application thereof, and pharmaceutical composition 国科温州研究院(温州生物材料与工程研究所) 2023-03-14 CN claimed
CN-115784987-A Compound related to pneumonia, preparation method and application thereof, and pharmaceutical composition 国科温州研究院(温州生物材料与工程研究所) 2023-03-14 CN disclosed
CN-108948014-A 1- aryl -4- Oxy-1, the preparation and application of the pyrido heterocycle compound of 4- dihydroquinoline structure 江西科技师范大学 2018-12-07 CN disclosed
EP-2799437-B1 QUINOLINE AND CINNOLINE DERIVATIVES AND USE THEREOF UNIV SHENYANG PHARMACEUTICAL (CN) 2016-09-14 EP disclosed
US-9382232-B2 Quinoline and cinnoline derivatives and their applications SHENYANG PHARMACEUTICAL UNIVERSITY (CN) 2016-07-05 US disclosed
US-20140364431-A1 Quinoline and cinnoline derivatives and their applications SHENYANG PHARMACEUTICAL UNIVERSITY (CN) 2014-12-11 US disclosed
EP-2799437-A1 QUINOLINE AND CINNOLINE COMPOUNDS AND USE THEREOF Shenyang Pharmaceutical University (CN) 2014-11-05 EP disclosed
EP-0360258-A2 Amino acid quinoline and naphthyridine derivatives ABBOTT LABORATORIES (US) 1990-03-28 EP disclosed
EP-0251308-A1 4-Quinolone-3-carboxylic-acid derivatives, process for their synthesis and pharmaceutical preparations containing them Chemie Linz Gesellschaft m.b.H. (AT) 1988-01-07 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20140364431-A1 Quinoline and cinnoline derivatives and their applications MET, CHEK1, KIT LMNA 1240/4885KDM4E 2948/4885MEN1 10/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.