SCHEMBL1044762

SCHEMBL1044762

O=C(O)N1CCC(CCC2(C(=O)OCc3ccccc3)CCCC2O)CC1

nearest known ligand 0.42

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 3/20 0.42
RAB9A P51151 2/20 0.42
NPC1 O15118 1/20 0.42
CYP2C19 P33261 1/20 0.41
GRIN2B Q13224 3/20 0.40
FAAH O00519 1/20 0.39
CYP2D6 P10635 1/20 0.39
CYP2C9 P11712 1/20 0.39
ALDH1A1 P00352 1/20 0.39
LMNA P02545 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3782495 0.93 SMN1; SMN2 (0.52) SMN1; SMN2RAB9ANPC1CYP2C19GRIN2B
SCHEMBL1043158 0.89 SMN1; SMN2 (0.44) SMN1; SMN2RAB9ANPC1CYP2C19GRIN2B
SCHEMBL1042956 0.84 NPC1 (0.38) SMN1; SMN2RAB9ANPC1
SCHEMBL3776399 0.82 SMN1; SMN2 (0.54) SMN1; SMN2RAB9ANPC1CYP2C19GRIN2B
SCHEMBL3788783 0.77 SMN1; SMN2 (0.46) SMN1; SMN2RAB9ANPC1CYP2C19GRIN2B
SCHEMBL3779088 0.77 DDB1 (0.39) SMN1; SMN2RAB9ANPC1CYP2C19CYP2C9
SCHEMBL3776673 0.77 CPB2 (0.40) SMN1; SMN2CYP2C19
SCHEMBL3787665 0.74 KCNA5 (0.42) SMN1; SMN2CYP2C19GRIN2BCYP2D6CYP2C9
SCHEMBL3781275 0.71 CYP17A1 (0.49) GRIN2BCYP2D6CYP2C9LMNA
SCHEMBL22117759 0.71 CHRM4 (0.49) SMN1; SMN2RAB9ANPC1CYP2C19GRIN2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2272826-A1 2-mercaptopentancarboxylic acid derivatives, the method for preparing them and the pharmaceutical compositions containing them Les Laboratoires Servier (FR) 2011-01-12 EP disclosed
WO-2010149888-A1 DERIVATIVES OF 2-MERCAPTOCYCLOPENTANE CARBOXYLIC ACID, METHOD FOR THE PREPARATION THEREOF, AND PHARMACEUTICAL COMPOSITIONS CONTAINING THE SAME LES LABORATOIRES SERVIER (FR) 2010-12-29 WO disclosed