SCHEMBL1045328

SCHEMBL1045328

CC1=NC=C[N+]1(Cc1ccccc1)Cc1ccccc1

nearest known ligand 0.38

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 1/20 0.38
TP53 P04637 1/20 0.33
HIF1A Q16665 1/20 0.32
TSHR P16473 3/20 0.32
KDM4E B2RXH2 2/20 0.31
CALM1 P0DP23 1/20 0.31
POLB P06746 1/20 0.31
ALDH1A1 P00352 1/20 0.30
NPSR1 Q6W5P4 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL10695236 0.98 CYP2D6 (0.37) CYP2D6TP53HIF1ATSHRKDM4E
SCHEMBL869872 0.61 TP53 (0.33) CYP2D6TP53HIF1ATSHRCALM1
SCHEMBL149879 0.58
SCHEMBL627768 0.57
SCHEMBL231005 0.57 ESR1 (0.56) TP53TSHRKDM4ECALM1ALDH1A1
SCHEMBL13326546 0.56 HIF1A (0.58) CYP2D6TP53HIF1ATSHRCALM1
SCHEMBL1017459 0.56 HIF1A (0.46) CYP2D6TP53HIF1ATSHRCALM1
Hydrochloric Acid SCHEMBL11729334 0.54 HIF1A (0.56) CYP2D6TP53HIF1ATSHRKDM4E
SCHEMBL6420860 0.54 TDP1 (0.52) TP53ALDH1A1
Toluene SCHEMBL4307944 0.54 LMNA (0.58) TP53TSHRKDM4ECALM1POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2803356-A1 Method for treating neurological disorders with imidazolium and imidazolinium compounds Agency for Science, Technology and Research (SG) 2014-11-19 EP disclosed
US-20110028513-A1 METHOD FOR TREATING NEUROLOGICAL DISORDERS WITH IMIDAZOLIUM AND IMIDAZOLINIUM COMPOUNDS AGENCY FOR SCIENCE, TECHNOLOGY AND RESEARCH (SG) 2011-02-03 US disclosed
EP-2271338-A1 METHOD FOR TREATING NEUROLOGICAL DISORDERS WITH IMIDAZOLIUM AND IMIDAZOLINIUM COMPOUNDS Agency for Science, Technology And Research (SG) 2011-01-12 EP disclosed
WO-2009123569-A1 METHOD FOR TREATING NEUROLOGICAL DISORDERS WITH IMIDAZOLIUM AND IMIDAZOLINIUM COMPOUNDS AGENCY FOR SCIENCE, TECHNOLOGY AND RESEARCH (SG) 2009-10-08 WO disclosed
EP-1337511-A1 BIS-HETEROCYCLIC COMPOUNDS WITH ANTITUMOUR AND CHEMOSENSITISING ACTIVITY Sigma-Tau Industrie Farmaceutiche Riunite S.p.A. (IT) 2003-08-27 EP disclosed
WO-2002036561-A1 BIS-HETEROCYCLIC COMPOUNDS WITH ANTITUMOUR AND CHEMOSENSITISING ACTIVITY SIGMA-TAU INDUSTRIE FARMACEUTICHE RIUNITE S.P.A. (IT) 2002-05-10 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110028513-A1 METHOD FOR TREATING NEUROLOGICAL DISORDERS WITH IMIDAZOLIUM AND IMIDAZOLINIUM COMPOUNDS SMN1; SMN2, INA, NLN CYP2D6 4802/4885TP53 3528/4885HIF1A 3823/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.