SCHEMBL10459592

SCHEMBL10459592

COCOc1cc2c(cc1Br)OCC2

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 3/20 0.34
HTR2C P28335 3/20 0.34
HTR2B P41595 2/20 0.34
HTR1A P08908 4/20 0.33
SLC6A4 P31645 4/20 0.33
CYP3A4 P08684 1/20 0.32
CYP2D6 P10635 1/20 0.32
CYP2C9 P11712 1/20 0.32
CYP2C19 P33261 1/20 0.32
DRD2 P14416 1/20 0.32
DRD3 P35462 1/20 0.32
MAPT P10636 2/20 0.32
HPGD P15428 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
NPSR1 Q6W5P4 1/20 0.32
TDP1 Q9NUW8 1/20 0.32
ERN1 O75460 1/20 0.32
CXCR3 P49682 1/20 0.31
P2RX7 Q99572 1/20 0.31
KDM4E B2RXH2 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20562373 0.84 MAPT (0.39) HTR1ASLC6A4CYP3A4CYP2D6CYP2C9
SCHEMBL5722666 0.82 HTR2C (0.50) HTR2AHTR2CHTR2BCYP3A4MAPT
SCHEMBL10460364 0.80 CXCR3 (0.33) HTR2AHTR2CCXCR3
SCHEMBL8323266 0.78 ERN1 (0.44) CYP3A4CYP2D6CYP2C9CYP2C19MAPT
SCHEMBL8133665 0.78 CYP3A4 (0.44) CYP3A4CYP2D6CYP2C9CYP2C19MAPT
SCHEMBL10459615 0.77 ERN1 (0.32) ERN1CXCR3
SCHEMBL10459591 0.77 HTR2A (0.33) HTR2AHTR2CHTR2BDRD2DRD3
SCHEMBL30665872 0.76 HTR2A (0.50) HTR2AHTR2CHTR2BERN1
SCHEMBL26654718 0.76 HTR2A (0.50) HTR2AHTR2CHTR2BERN1
SCHEMBL10459600 0.74 CLK1 (0.43) CYP3A4CYP2D6CYP2C9CYP2C19MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4966907-A ANTIINFLAMMATORY AGENT, ANTIALLERGENS MERCK & CO., INC. (US) 1990-10-30 US disclosed