SCHEMBL10463551

SCHEMBL10463551

Cc1cc(-n2cnnn2)ccc1N

nearest known ligand 0.62

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.57
MAPT P10636 3/20 0.57
LMNA P02545 2/20 0.57
HTT P42858 1/20 0.57
NOTUM Q6P988 7/20 0.53
F2 P00734 1/20 0.49
KCNJ1 P48048 2/20 0.47
KDM4E B2RXH2 1/20 0.45
RAD52 P43351 1/20 0.45
TP53 P04637 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17725782 0.84 ALDH1A1 (0.62) ALDH1A1MAPTLMNAHTTNOTUM
SCHEMBL24769728 0.84 NOTUM (0.58) ALDH1A1MAPTLMNAHTTNOTUM
SCHEMBL1577735 0.79 MAPT (0.58) ALDH1A1MAPTLMNAHTTNOTUM
SCHEMBL22637227 0.79 NOTUM (0.53) ALDH1A1MAPTLMNAHTTNOTUM
SCHEMBL24073776 0.79 NOTUM (0.53) ALDH1A1MAPTLMNAHTTNOTUM
SCHEMBL15872005 0.79 NOTUM (0.72) ALDH1A1MAPTLMNAHTTNOTUM
SCHEMBL24073780 0.79 NOTUM (0.49) ALDH1A1MAPTLMNAHTTNOTUM
SCHEMBL221145 0.79 ALDH1A1 (0.56) ALDH1A1MAPTLMNAHTTNOTUM
SCHEMBL24073374 0.78 NOTUM (0.47) ALDH1A1MAPTLMNAHTTNOTUM
SCHEMBL19398295 0.77 ALDH1A1 (0.54) ALDH1A1MAPTLMNAHTTNOTUM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012129452-A2 PROPYNOIC ACID CARBAMOYL METHYL-ALMIDES AND PHARMACEUTICAL COMPOSITIONS AND METHODS BASED THEREON UNIVERSITY OF SOUTHERN CALIFORNIA (US) 2012-09-27 WO disclosed
US-4900839-A SUBSTITUTED PHENYLPROPENAMIDES PFIZER INC. (US) 1990-02-13 US disclosed
US-4837334-A Precursors to quinolone inotropic agents PFIZER INC. (US) 1989-06-06 US disclosed
US-4728653-A CONGESTIVE HEART FAILURE PFIZER INC. (US) 1988-03-01 US disclosed