SCHEMBL10463602

SCHEMBL10463602

CC1CC(=O)NN=C1c1ccc2[nH]c(-c3ccccn3)nc2c1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE3B Q13370 8/20 0.57
PDE3A Q14432 8/20 0.57
ABCB11 O95342 1/20 0.56
MAOA P21397 1/20 0.56
ADORA2A P29274 1/20 0.56
F10 P00742 1/20 0.53
GPR119 Q8TDV5 6/20 0.50
NPC1 O15118 2/20 0.50
LMNA P02545 2/20 0.50
PKM P14618 2/20 0.50
RAB9A P51151 2/20 0.50
SMN1; SMN2 Q16637 2/20 0.50
KDM4E B2RXH2 1/20 0.50
MAPT P10636 1/20 0.50
KMT2A Q03164 1/20 0.50
METAP2 P50579 2/20 0.48
METAP1 P53582 2/20 0.48
CBFB Q13951 2/20 0.48
PDE4A P27815 2/20 0.47
PDE4B Q07343 2/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL9781443 0.98 PDE3B (0.56) PDE3BPDE3AABCB11MAOAADORA2A
SCHEMBL10463603 0.92 PDE3B (0.68) PDE3BPDE3AABCB11MAOAADORA2A
Hydrochloric Acid SCHEMBL9781446 0.90 PDE3B (0.66) PDE3BPDE3AABCB11MAOAADORA2A
SCHEMBL10922000 0.88 PDE3B (0.56) PDE3BPDE3AABCB11MAOAADORA2A
SCHEMBL10774240 0.84 F10 (0.55) PDE3BPDE3AABCB11MAOAADORA2A
SCHEMBL9781454 0.84 PDE3B (0.64) PDE3BPDE3AABCB11MAOAADORA2A
Meribendan SCHEMBL9781483 0.83 PDE3B (0.58) PDE3BPDE3AABCB11MAOAADORA2A
SCHEMBL29698511 0.83 GPR119 (0.54) PDE3BPDE3AGPR119PDE4APDE4B
SCHEMBL10769306 0.83 PDE3B (0.60) PDE3BPDE3AABCB11MAOAADORA2A
SCHEMBL10770212 0.82 PDE3B (0.57) PDE3BPDE3AABCB11MAOAADORA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4923869-A INOTROPIC, VASODILATING, AND ANTITHROMBOTIC AGENTS MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1990-05-08 US claimed
EP-0193013-B1 BENZIMIDAZOLYL-PYRIDAZINONES MERCK PATENT GmbH (DE) 1989-04-19 EP claimed
EP-0193013-B1 BENZIMIDAZOLYL-PYRIDAZINONES MERCK PATENT GmbH (DE) 1989-04-19 EP disclosed