SCHEMBL10465331

SCHEMBL10465331

CC(C)(Cc1ccc(SC(F)(F)F)cc1)C(=O)c1cncnc1

nearest known ligand 0.44

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
EPHX2 P34913 1/20 0.44
NR1H4 Q96RI1 1/20 0.44
NTRK1 P04629 2/20 0.41
PTPRZ1 P23471 4/20 0.41
KDM4E B2RXH2 1/20 0.39
ALDH1A1 P00352 1/20 0.39
TDP1 Q9NUW8 1/20 0.39
ABL1 P00519 4/20 0.39
PTPN1 P18031 2/20 0.39
TRPV1 Q8NER1 1/20 0.39
KIF11 P52732 1/20 0.36
MBOAT4 Q96T53 1/20 0.34
LMNA P02545 1/20 0.34
MAPT P10636 1/20 0.34
TSHR P16473 1/20 0.34
MAPK1 P28482 1/20 0.34
HTT P42858 1/20 0.34
KCNH2 Q12809 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10465612 0.82 CYP19A1 (0.40) NTRK1PTPN1TRPV1LMNAHTT
SCHEMBL10464161 0.82 CXCR4 (0.39) NTRK1KDM4EALDH1A1ABL1TSHR
SCHEMBL10518546 0.79 SLC6A2 (0.46) NTRK1LMNAMAPTTSHR
SCHEMBL10465337 0.77 EPHX2 (0.49) EPHX2NR1H4PTPRZ1KDM4EALDH1A1
SCHEMBL10465910 0.74 PTPRZ1 (0.39) EPHX2NR1H4NTRK1PTPRZ1KDM4E
SCHEMBL9203686 0.72 CYP3A4 (0.41) EPHX2NR1H4PTPRZ1ALDH1A1PTPN1
SCHEMBL10465335 0.71 EPHX2 (0.44) EPHX2NR1H4PTPRZ1KDM4EALDH1A1
SCHEMBL13020828 0.69 PTPRZ1 (0.57) EPHX2NR1H4PTPRZ1KDM4EALDH1A1
SCHEMBL9790519 0.68 HCAR2 (0.45) KDM4ETDP1LMNA
SCHEMBL10585982 0.68 SMN1; SMN2 (0.40) ALDH1A1MAPTKCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4939155-A Fungicides BAYER AKTIENGESELLSCHAFT (DE) 1990-07-03 US disclosed
US-4877446-A FUNGICIDES BAYER AKTIENGESELLSCHAFT (DE) 1989-10-31 US disclosed
EP-0277520-A2 Parasiticide on a pyrimidine derivative basis BAYER AG (DE) 1988-08-10 EP disclosed