SCHEMBL10470951

SCHEMBL10470951

CC#CCN1CCCC1=O

nearest known ligand 0.66

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CHRM2 P08172 5/20 0.65
CHRM5 P08912 5/20 0.65
CHRM1 P11229 5/20 0.65
CHRM3 P20309 4/20 0.65
CYP2D6 P10635 2/20 0.65
CHRM4 P08173 2/20 0.65
CYP1A2 P05177 1/20 0.65
CYP2C9 P11712 1/20 0.65
CYP2C19 P33261 1/20 0.65
ALDH1A1 P00352 2/20 0.64
LMNA P02545 2/20 0.64
APEX1 P27695 2/20 0.64
PMP22 Q01453 2/20 0.64
TSHR P16473 1/20 0.64
ALOX12 P18054 1/20 0.64
NFKB1 P19838 1/20 0.64
MAPK1 P28482 1/20 0.64

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3021293 0.82 CHRM2 (0.50) CHRM2CHRM5CHRM1CHRM3CYP2D6
SCHEMBL12004137 0.82 CHRM2 (0.67) CHRM2CHRM5CHRM1CHRM3CYP2D6
SCHEMBL9468715 0.80 CHRM2 (0.65) CHRM2CHRM5CHRM1CHRM3CYP2D6
SCHEMBL9029739 0.78 CHRM2 (0.68) CHRM2CHRM5CHRM1CHRM3CYP2D6
Oxotremorine SCHEMBL2128 0.78 CHRM2 (1.00) CHRM2CHRM5CHRM1CHRM3CYP2D6
Hydrochloric Acid SCHEMBL7371622 0.78 CHRM2 (0.62) CHRM2CHRM5CHRM1CHRM3CYP2D6
SCHEMBL31263727 0.78 CHRM2 (0.93) CHRM2CHRM5CHRM1CHRM3CYP2D6
SCHEMBL11725908 0.78 CHRM2 (0.62) CHRM2CHRM5CHRM1CHRM3CYP2D6
Oxotremorine SCHEMBL1320883 0.78 CHRM2 (0.90) CHRM2CHRM5CHRM1CHRM3CYP2D6
SCHEMBL4542695 0.78 CHRM2 (1.00) CHRM2CHRM5CHRM1CHRM3CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7825155-B2 Oxindole derivative as feeding control agent DAINIPPON SUMITOMO PHARMA CO., LTD. (JP) 2010-11-02 US disclosed
US-20090131398-A1 OXINDOLE DERIVATIVE AS FEEDING CONTROL AGENT DAINIPPON SUMITOMO PHARMA CO., LTD. (JP) 2009-05-21 US disclosed
US-4916139-A TREATMENT OF CONVULSIONS, DEPRESSION, HYPERTENSION, PAIN HOECHST-ROUSSEL PHARMACEUTICALS, INC. (US) 1990-04-10 US disclosed
EP-0333026-A1 3-(2,3,4,5,6-Pentafluorophenoxy)-8-azabicyclo[3.2.1]octanes, a process for their preparation and their use as medicaments HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1989-09-20 EP disclosed
US-4861889-A 3-(2,3,4,5,6-pentafluorophenoxy)-8-azabicyclo[3.2.1]octanes HOECHST-ROUSSEL PHARMACEUTICALS, INC. (US) 1989-08-29 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090131398-A1 OXINDOLE DERIVATIVE AS FEEDING CONTROL AGENT GPR119, OXTR, CCKAR CHRM2 151/4885CHRM5 314/4885CHRM1 95/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.