SCHEMBL10474199

SCHEMBL10474199

CCCCCNc1ccc(C2=NNC(=O)CC2)cc1

nearest known ligand 0.66

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 2/20 0.62
NPY1R P25929 1/20 0.62
NPY2R P49146 1/20 0.62
MAPT P10636 2/20 0.55
KCNH2 Q12809 1/20 0.54
SMN1; SMN2 Q16637 1/20 0.50
PDE3B Q13370 10/20 0.46
PDE3A Q14432 9/20 0.46
KMT2A Q03164 1/20 0.46
PDE2A O00408 1/20 0.46
PDE1A P54750 1/20 0.46
PDE1B Q01064 1/20 0.46
PDE1C Q14123 1/20 0.46
PDE4A P27815 4/20 0.45
PDE4B Q07343 4/20 0.45
PDE4C Q08493 4/20 0.45
PDE4D Q08499 4/20 0.45
CYP1A2 P05177 1/20 0.45
CYP3A4 P08684 1/20 0.45
CYP2D6 P10635 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10463523 0.86 KCNH2 (0.53) LMNANPY1RNPY2RMAPTKCNH2
SCHEMBL10465918 0.85 KCNH2 (0.56) LMNANPY1RNPY2RMAPTKCNH2
SCHEMBL21970671 0.85 KCNH2 (0.61) LMNANPY1RNPY2RMAPTKCNH2
SCHEMBL10464834 0.79 LMNA (0.50) LMNANPY1RNPY2RMAPTKCNH2
SCHEMBL9815919 0.78 LMNA (0.65) LMNANPY1RNPY2RMAPTKCNH2
SCHEMBL10464942 0.78 LMNA (0.52) LMNANPY1RNPY2RMAPTKCNH2
SCHEMBL22910067 0.77 KCNH2 (0.66) LMNANPY1RNPY2RMAPTKCNH2
SCHEMBL10619654 0.77 LMNA (0.47) LMNANPY1RNPY2RMAPTSMN1; SMN2
SCHEMBL10967326 0.77 LMNA (1.00) LMNANPY1RNPY2RMAPTKCNH2
SCHEMBL10464826 0.77 LMNA (0.45) LMNANPY1RNPY2RMAPTKCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 17 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0042107-B1 DIHYDROPYRIDAZINONES, PROCESSES FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THESE COMPOUNDS BASF Aktiengesellschaft (DE) 1985-04-03 EP claimed
US-4410529-A HYPOTENSIVE AGNENTS, ANTICOAGULANTS BASF AKTIENGESELLSCHAFT (DE) 1983-10-18 US claimed
EP-0042107-A1 Dihydropyridazinones, processes for their preparation and pharmaceutical compositions containing these compounds BASF Aktiengesellschaft (DE) 1981-12-23 EP claimed
EP-0012338-A1 Dihydropyridazinones, process for their preparation and therapeutical agents containing them BASF Aktiengesellschaft (DE) 1980-06-25 EP claimed
US-4965263-A HYPOTENSIVE AGENTS MITSUI TOATSU KAGAKU KABUSHIKI KAISHA (JP) 1990-10-23 US disclosed
EP-0090978-B1 IMIDAZOLYLPHENYL-TETRAHYDROPYRIDAZINES, PROCESS FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM A. Nattermann & Cie. GmbH (DE) 1988-11-30 EP disclosed
EP-0107735-B1 NOVEL PYRIDAZINONE DERIVATIVES MITSUI TOATSU KAGAKU KABUSHIKI KAISHA (JP) 1988-10-19 EP disclosed
US-4639451-A HYPOTENSIVE AGENTS, ANTICOAGULANTS MITSUI TOATSU KAGAKU-KABUSHIKI KAISHA (JP) 1987-01-27 US disclosed
EP-0042107-B1 DIHYDROPYRIDAZINONES, PROCESSES FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THESE COMPOUNDS BASF Aktiengesellschaft (DE) 1985-04-03 EP disclosed
EP-0107735-A1 NOVEL PYRIDAZINONE DERIVATIVES MITSUI TOATSU KAGAKU KABUSHIKI KAISHA (JP) 1984-05-09 EP disclosed
US-4410529-A HYPOTENSIVE AGNENTS, ANTICOAGULANTS BASF AKTIENGESELLSCHAFT (DE) 1983-10-18 US disclosed
US-4410529-A HYPOTENSIVE AGNENTS, ANTICOAGULANTS BASF AKTIENGESELLSCHAFT (DE) 1983-10-18 US disclosed
EP-0090978-A2 Imidazolylphenyl-tetrahydropyridazines, process for their preparation and pharmaceutical compositions containing them A. Nattermann & Cie. GmbH (DE) 1983-10-12 EP disclosed
EP-0042107-A1 Dihydropyridazinones, processes for their preparation and pharmaceutical compositions containing these compounds BASF Aktiengesellschaft (DE) 1981-12-23 EP disclosed
EP-0042107-A1 Dihydropyridazinones, processes for their preparation and pharmaceutical compositions containing these compounds BASF Aktiengesellschaft (DE) 1981-12-23 EP disclosed
EP-0012338-A1 Dihydropyridazinones, process for their preparation and therapeutical agents containing them BASF Aktiengesellschaft (DE) 1980-06-25 EP disclosed
EP-0012338-A1 Dihydropyridazinones, process for their preparation and therapeutical agents containing them BASF Aktiengesellschaft (DE) 1980-06-25 EP disclosed