SCHEMBL10474227

SCHEMBL10474227

Cc1ccc(C)n1NC(=O)COc1ccc(C2=NNC(=O)CC2)cc1Cl

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 3/20 0.52
MEN1 O00255 2/20 0.52
PDE3B Q13370 8/20 0.47
PDE3A Q14432 8/20 0.47
PDE4B Q07343 4/20 0.47
PDE4A P27815 3/20 0.47
PDE4C Q08493 3/20 0.47
PDE4D Q08499 3/20 0.47
MAPT P10636 5/20 0.41
TP53 P04637 1/20 0.41
GAA P10253 1/20 0.41
HPGD P15428 1/20 0.41
LMNA P02545 3/20 0.41
NPY1R P25929 1/20 0.41
NPY2R P49146 1/20 0.41
ALDH1A1 P00352 3/20 0.39
TSHR P16473 1/20 0.39
MAPK1 P28482 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
HRH3 Q9Y5N1 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10474304 0.83 PDE3B (0.50) KMT2APDE3BPDE3APDE4BPDE4A
SCHEMBL9657441 0.82 PDE3B (0.47) KMT2APDE3BPDE3APDE4BPDE4A
SCHEMBL10867608 0.81 PDE4B (0.48) KMT2APDE3BPDE3APDE4BPDE4A
SCHEMBL4573757 0.81 PDE3B (0.54) KMT2APDE3BPDE3APDE4BPDE4A
SCHEMBL4573518 0.81 PDE3B (0.52) KMT2AMEN1PDE3BPDE3APDE4B
SCHEMBL9526509 0.80 LMNA (0.51) KMT2APDE3BPDE3APDE4BPDE4A
SCHEMBL9657454 0.80 PDE3B (0.45) KMT2APDE3BPDE3APDE4BPDE4A
SCHEMBL7337123 0.80 PDE3B (0.46) PDE3BPDE3APDE4BPDE4APDE4C
SCHEMBL10475455 0.80 HPGD (0.49) KMT2APDE3BPDE3APDE4BPDE4A
SCHEMBL7326426 0.80 PDE3B (0.47) KMT2APDE3BPDE3APDE4BPDE4A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4914093-A CARDIOVASCULAR DISORDERS SANKYO COMPANY LIMITED (JP) 1990-04-03 US disclosed
EP-0330242-A1 Pyridazinone derivatives, their preparation and use Sankyo Company Limited (JP) 1989-08-30 EP disclosed
EP-0178189-A2 Pyridazinone derivatives, their preparation and use SANKYO COMPANY LIMITED (JP) 1986-04-16 EP disclosed