SCHEMBL10476325

SCHEMBL10476325

O=C(NCc1ccc(C(F)(F)F)cc1)c1ccc(CSc2c(Cl)ccc3c2CCNCC3)cc1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LSS P48449 1/20 0.43
MAPK14 Q16539 1/20 0.42
CHRM3 P20309 1/20 0.42
NAMPT P43490 1/20 0.41
EPHX2 P34913 3/20 0.40
PPARG P37231 2/20 0.40
PPARA Q07869 1/20 0.40
MAOA P21397 1/20 0.39
MEN1 O00255 2/20 0.39
CYP1A2 P05177 2/20 0.39
CYP2C19 P33261 2/20 0.39
KMT2A Q03164 2/20 0.39
PSMD14 O00487 1/20 0.38
STAMBP O95630 1/20 0.38
POLB P06746 1/20 0.38
CYP3A4 P08684 1/20 0.38
CYP2D6 P10635 1/20 0.38
CYP2C9 P11712 1/20 0.38
HPGD P15428 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL507842 0.99 LSS (0.43) LSSMAPK14CHRM3NAMPTEPHX2
SCHEMBL10476134 0.94 MLYCD (0.47) LSSMAPK14CHRM3NAMPTEPHX2
SCHEMBL508437 0.91 LMNA (0.49) PPARGPOLBSMN1; SMN2HDAC1HDAC4
SCHEMBL10476163 0.89 EPHX2 (0.40) CHRM3EPHX2PPARGPPARAKMT2A
SCHEMBL10476267 0.86 PPARG (0.45) CHRM3EPHX2PPARGHDAC1HDAC4
Hydrochloric Acid SCHEMBL507616 0.85 PPARG (0.44) CHRM3EPHX2PPARGHDAC1HDAC4
Succinic Acid SCHEMBL507971 0.85 PPARD (0.38) CHRM3EPHX2PPARGPPARAKMT2A
SCHEMBL10476291 0.85 EPHX2 (0.47) EPHX2PPARGPPARA
SCHEMBL10476165 0.84 HTR2C (0.37) LSSMEN1KMT2ACYP3A4CYP2D6
SCHEMBL10278060 0.84 MEN1 (0.39) NAMPTMEN1CYP1A2CYP2C19KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8580780-B2 6 substituted 2, 3,4,5 tetrahydro-1H-benzo[d]azepines as 5-HT2C receptor agonist ELI LILLY AND COMPANY (US) 2013-11-12 US claimed
EP-2479168-A1 6-Substituted 2,3,4,5-Tetrahydro-1H-Benzo [d]Azepines as 5-HT2C Receptor Agonists ELI LILLY AND COMPANY (US) 2012-07-25 EP claimed