SCHEMBL10479481

SCHEMBL10479481

O=C(O)c1nn(-c2ccc(Cl)cc2)c2c1CCC2

nearest known ligand 0.57

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 8/20 0.57
PTGS1 P23219 4/20 0.57
CYP1A2 P05177 3/20 0.47
HIF1A Q16665 1/20 0.47
GRIA2 P42262 3/20 0.46
CYP2C9 P11712 1/20 0.46
UGCG Q16739 2/20 0.46
CNR1 P21554 1/20 0.46
CNR2 P34972 1/20 0.46
GAA P10253 1/20 0.45
FABP4 P15090 1/20 0.44
CYP2C19 P33261 1/20 0.44
RPA1 P27694 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
CYP2D6 P10635 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5812502 0.97 PTGS2 (0.59) PTGS2PTGS1CYP1A2HIF1AGRIA2
SCHEMBL20604173 0.86 PTGS2 (0.60) PTGS2PTGS1CYP1A2GRIA2CYP2C9
SCHEMBL10479480 0.85 GRIA2 (0.46) PTGS2PTGS1CYP1A2GRIA2CYP2C9
SCHEMBL14662754 0.83 PTGS2 (0.60) PTGS2PTGS1CYP1A2GRIA2CYP2C9
SCHEMBL10479738 0.82 GRIA2 (0.46) PTGS2PTGS1CYP1A2GRIA2CYP2C9
SCHEMBL25434903 0.82 TP53 (0.55) PTGS2PTGS1UGCGFABP4RPA1
SCHEMBL5811399 0.82 CNR1 (0.65) PTGS2UGCGCNR1CNR2RPA1
SCHEMBL10479510 0.81 KDM4E (0.49) PTGS2CYP1A2GRIA2CYP2C9GAA
SCHEMBL10479625 0.80 KMT2A (0.54) PTGS2PTGS1SMN1; SMN2
SCHEMBL10479406 0.79 PTGS2 (0.58) PTGS2PTGS1CYP1A2GRIA2CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4851425-A Cyclopentapyrazole and tetrahydroindazole compounds and their use as anti-inflammatory and anti-allergic agents THE UPJOHN COMPANY (US) 1989-07-25 US disclosed