SCHEMBL5812502

SCHEMBL5812502

O=C(O)c1nn(-c2ccc(Cl)cc2)c2c1CCCC2

nearest known ligand 0.59

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 8/20 0.59
PTGS1 P23219 6/20 0.57
GRIA2 P42262 7/20 0.49
CYP1A2 P05177 3/20 0.49
CYP2C9 P11712 3/20 0.49
CNR1 P21554 1/20 0.48
CNR2 P34972 1/20 0.48
GAA P10253 1/20 0.48
CYP2C19 P33261 1/20 0.47
HIF1A Q16665 1/20 0.47
CYP2D6 P10635 2/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10479481 0.97 PTGS2 (0.57) PTGS2PTGS1GRIA2CYP1A2CYP2C9
SCHEMBL14662754 0.86 PTGS2 (0.60) PTGS2PTGS1GRIA2CYP1A2CYP2C9
SCHEMBL10479738 0.85 GRIA2 (0.46) PTGS2PTGS1GRIA2CYP1A2CYP2C9
SCHEMBL5811399 0.85 CNR1 (0.65) PTGS2CNR1CNR2
SCHEMBL20604173 0.83 PTGS2 (0.60) PTGS2PTGS1GRIA2CYP1A2CYP2C9
SCHEMBL10479480 0.82 GRIA2 (0.46) PTGS2PTGS1GRIA2CYP1A2CYP2C9
SCHEMBL10479406 0.82 PTGS2 (0.58) PTGS2PTGS1GRIA2CYP1A2CYP2C9
SCHEMBL10479633 0.81 KDM4E (0.49) PTGS2PTGS1GRIA2CYP1A2CYP2C9
SCHEMBL5810803 0.81 OPRM1 (0.52) CNR1CNR2
SCHEMBL4219942 0.81 PTGS2 (0.60) PTGS2PTGS1GRIA2CYP1A2CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2006030124-A1 CONDENSED PYRAZOLE DERIVATIVES, PREPARATION METHOD THEREOF AND THERAPEUTIC USE OF SAME SANOFI-AVENTIS (FR) 2006-03-23 WO disclosed
US-4851425-A Cyclopentapyrazole and tetrahydroindazole compounds and their use as anti-inflammatory and anti-allergic agents THE UPJOHN COMPANY (US) 1989-07-25 US disclosed
WO-1986007357-A3 CYCLOPENTAPYRAZOLE AND TETRAHYDROINDAZOLE COMPOUNDS THE UPJOHN COMPANY (US) 1987-04-23 WO disclosed