SCHEMBL10487948

SCHEMBL10487948

O=c1[nH]c2ccccc2c(=O)n1Cc1ccc(Br)cc1F

nearest known ligand 0.58

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.58
HPGD P15428 3/20 0.58
KDM4E B2RXH2 3/20 0.58
SMN1; SMN2 Q16637 1/20 0.58
HSP90AA1 P07900 2/20 0.54
TRAP1 Q12931 2/20 0.53
HSP90B1 P14625 1/20 0.53
OPRM1 P35372 1/20 0.53
CYP1A2 P05177 2/20 0.52
TSHR P16473 1/20 0.51
MEN1 O00255 4/20 0.48
KMT2A Q03164 4/20 0.48
DDR1 Q08345 2/20 0.47
HSD17B10 Q99714 2/20 0.47
AKR1B1 P15121 2/20 0.47
CYP2C9 P11712 1/20 0.47
MAPK1 P28482 1/20 0.45
AKR1A1 P14550 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10487936 0.90 TRAP1 (0.55) ALDH1A1HPGDKDM4ESMN1; SMN2HSP90AA1
SCHEMBL10487983 0.86 TRAP1 (0.52) ALDH1A1HPGDKDM4ESMN1; SMN2HSP90AA1
SCHEMBL7752011 0.84 AKR1A1 (0.58) ALDH1A1HSP90AA1TRAP1HSP90B1OPRM1
SCHEMBL10487924 0.84 TRAP1 (0.53) ALDH1A1HPGDKDM4ESMN1; SMN2HSP90AA1
SCHEMBL10488205 0.82 TRAP1 (0.59) ALDH1A1SMN1; SMN2HSP90AA1TRAP1HSP90B1
SCHEMBL10487908 0.82 DDR1 (0.58) HSP90AA1TRAP1HSP90B1DDR1
SCHEMBL10487998 0.81 TRAP1 (0.47) ALDH1A1HPGDKDM4ESMN1; SMN2HSP90AA1
SCHEMBL10488017 0.79 TRAP1 (0.51) ALDH1A1KDM4ESMN1; SMN2HSP90AA1TRAP1
Acetic Acid SCHEMBL4363267 0.79 AKR1B1 (0.60) HPGDKDM4EHSP90AA1TRAP1HSP90B1
SCHEMBL7101724 0.76 KMT2A (0.78) ALDH1A1HPGDKDM4ESMN1; SMN2CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4883800-A DIABETES FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1989-11-28 US disclosed
US-4734419-A Quinazoline derivatives, compositions thereof and their use in treating diabetic complications FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1988-03-29 US disclosed
EP-0218999-A2 New quinazoline derivatives, process for their production and pharmaceutical compositions comprising them FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1987-04-22 EP disclosed