SCHEMBL10488134

SCHEMBL10488134

CCCOC(=O)c1ccc(C#CCCOCCCCCBr)cc1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 3/20 0.46
ALDH1A1 P00352 2/20 0.46
ESR1 P03372 2/20 0.46
CHRM1 P11229 1/20 0.46
SLC6A2 P23975 1/20 0.46
KDR P35968 1/20 0.46
TDP1 Q9NUW8 1/20 0.46
PTPN2 P17706 6/20 0.44
PTPN1 P18031 6/20 0.44
PTPN6 P29350 6/20 0.44
PTPN11 Q06124 6/20 0.44
NPC1 O15118 1/20 0.44
MAPT P10636 1/20 0.44
RAB9A P51151 1/20 0.44
LMNA P02545 3/20 0.43
MMP2 P08253 1/20 0.42
MMP12 P39900 1/20 0.42
CYP1A2 P05177 2/20 0.41
CYP2C19 P33261 2/20 0.41
CYP2D6 P10635 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10390471 0.81 PLA2G4B (0.54) TSHRALDH1A1ESR1CHRM1SLC6A2
SCHEMBL9763616 0.81 HRH3 (0.39) ALDH1A1NPC1MAPTRAB9ALMNA
SCHEMBL9763284 0.81 GPR119 (0.39) ALDH1A1PTPN2PTPN1PTPN6PTPN11
SCHEMBL9763014 0.79 ALDH1A1 (0.51) TSHRALDH1A1ESR1CHRM1SLC6A2
SCHEMBL9763584 0.79 ALDH1A1 (0.51) TSHRALDH1A1ESR1CHRM1SLC6A2
SCHEMBL10488165 0.76 CYP3A4 (0.36) PTPN2PTPN1PTPN6PTPN11MMP2
SCHEMBL10464556 0.75 PTPN2 (0.40) CHRM1PTPN2PTPN1PTPN6PTPN11
SCHEMBL17350477 0.75 ALDH1A1 (0.69) TSHRALDH1A1ESR1NPC1MAPT
SCHEMBL10488159 0.74 AR (0.45) ALDH1A1KDRNPC1RAB9ALMNA
SCHEMBL31284746 0.74 TSHR (0.56) TSHRALDH1A1ESR1NPC1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4853382-A TREATING ASTHMA AND BRONCHITIS GLAXO GROUP LIMITED (GB) 1989-08-01 US disclosed
EP-0178919-B1 AMINOPHENOL DERIVATIVES GLAXO GROUP LIMITED (GB) 1988-12-21 EP disclosed
US-4730008-A STIMULANT FOR BETA-ADRENORECEPTORS GLAXO GROUP LIMITED (GB) 1988-03-08 US disclosed