SCHEMBL10488255

SCHEMBL10488255

Cc1cc2c(Cl)c3ccccc3c(CNC(C)(CO)CO)c2cc1C

nearest known ligand 0.36

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
CD274 Q9NZQ7 1/20 0.36
SLC2A1 P11166 1/20 0.35
NPBWR1 P48145 1/20 0.34
KMT2A Q03164 1/20 0.34
MCHR1 Q99705 1/20 0.34
CYP1A2 P05177 1/20 0.33
MCL1 Q07820 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL10488357 0.99 CD274 (0.36) CD274SLC2A1NPBWR1KMT2AMCHR1
SCHEMBL10488837 0.90 KMT2A (0.38) CD274SLC2A1NPBWR1KMT2AMCHR1
Hydrochloric Acid SCHEMBL10488883 0.89 KMT2A (0.40) CD274SLC2A1NPBWR1KMT2AMCHR1
Hydrochloric Acid SCHEMBL10349542 0.88 NPBWR1 (0.40) CD274SLC2A1NPBWR1KMT2AMCHR1
SCHEMBL10488250 0.86 KMT2A (0.38) CD274SLC2A1NPBWR1KMT2AMCHR1
SCHEMBL10488373 0.86 SLC2A1 (0.40) CD274SLC2A1NPBWR1KMT2AMCHR1
Hydrochloric Acid SCHEMBL10488310 0.85 SLC2A1 (0.42) CD274SLC2A1NPBWR1KMT2AMCHR1
Hydrochloric Acid SCHEMBL10488570 0.85 KMT2A (0.40) CD274SLC2A1NPBWR1KMT2AMCHR1
SCHEMBL10488900 0.84 KIF11 (0.35) CD274SLC2A1NPBWR1KMT2AMCHR1
SCHEMBL10488323 0.84 KIF11 (0.35) CD274SLC2A1NPBWR1KMT2AMCHR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0125701-B1 POLYCYCLIC AROMATIC COMPOUNDS THE WELLCOME FOUNDATION LIMITED (GB) 1988-08-03 EP claimed
EP-0125701-A2 Polycyclic aromatic compounds THE WELLCOME FOUNDATION LIMITED (GB) 1984-11-21 EP claimed
US-4803226-A ANTITUMOR AGENTS BURROUGHS WELLCOME CO. (US) 1989-02-07 US disclosed
US-4803221-A Anthracene derivatives BURROUGHS WELLCOME CO. (US) 1989-02-07 US disclosed
EP-0125701-B1 POLYCYCLIC AROMATIC COMPOUNDS THE WELLCOME FOUNDATION LIMITED (GB) 1988-08-03 EP disclosed
US-4719047-A ANTITUMOR BURROUGHS WELLCOME CO. (US) 1988-01-12 US disclosed
US-4719049-A ANTITUMOR BURROUGHS WELLCOME CO. (US) 1988-01-12 US disclosed
EP-0125701-A2 Polycyclic aromatic compounds THE WELLCOME FOUNDATION LIMITED (GB) 1984-11-21 EP disclosed