SCHEMBL10488343

SCHEMBL10488343

CCc1ccc2cc3ccccc3c(CNC(C)(CO)CO)c2c1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 2/20 0.44
NPBWR1 P48145 1/20 0.44
MCHR1 Q99705 1/20 0.44
CYP1A2 P05177 1/20 0.41
CYP2A6 P11509 1/20 0.41
SLC2A1 P11166 1/20 0.39
HTR2A P28223 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.34
CNR2 P34972 2/20 0.33
CD274 Q9NZQ7 1/20 0.33
GAA P10253 1/20 0.33
POLB P06746 1/20 0.33
TP53 P04637 1/20 0.33
MEN1 O00255 1/20 0.33
ALDH1A1 P00352 1/20 0.33
CYP2D6 P10635 1/20 0.33
NCEH1 Q6PIU2 1/20 0.33
KIF11 P52732 1/20 0.33
SIGMAR1 Q99720 1/20 0.32
IDO1 P14902 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10488442 0.92 CYP1A2 (0.41) KMT2ANPBWR1MCHR1CYP1A2CYP2A6
SCHEMBL10488406 0.88 HTR2A (0.43) KMT2ANPBWR1MCHR1CYP1A2SLC2A1
Hydrochloric Acid SCHEMBL10488372 0.86 KMT2A (0.43) KMT2ANPBWR1MCHR1CYP1A2SLC2A1
SCHEMBL10348808 0.85 KMT2A (0.40) KMT2ANPBWR1MCHR1CYP1A2SLC2A1
SCHEMBL10488585 0.83 KMT2A (0.50) KMT2ANPBWR1MCHR1CYP1A2CYP2A6
Hydrochloric Acid SCHEMBL10488318 0.82 KMT2A (0.52) KMT2ANPBWR1MCHR1CYP1A2CYP2A6
SCHEMBL10348864 0.80 KMT2A (0.41) KMT2ANPBWR1MCHR1CYP1A2CYP2A6
SCHEMBL10488510 0.80 HTR2A (0.39) KMT2ANPBWR1MCHR1CYP1A2SLC2A1
SCHEMBL10348690 0.80 SLC2A1 (0.48) KMT2ANPBWR1MCHR1SLC2A1HTR2A
SCHEMBL1070224 0.79 CYP1A2 (0.52) CYP1A2CYP2A6HTR2AL3MBTL1CNR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0125702-B1 POLYCYCLIC AROMATIC COMPOUNDS THE WELLCOME FOUNDATION LIMITED (GB) 1987-08-12 EP claimed
US-4803221-A Anthracene derivatives BURROUGHS WELLCOME CO. (US) 1989-02-07 US disclosed
US-4719049-A ANTITUMOR BURROUGHS WELLCOME CO. (US) 1988-01-12 US disclosed
EP-0125702-B1 POLYCYCLIC AROMATIC COMPOUNDS THE WELLCOME FOUNDATION LIMITED (GB) 1987-08-12 EP disclosed
EP-0125702-A2 Polycyclic aromatic compounds THE WELLCOME FOUNDATION LIMITED (GB) 1984-11-21 EP disclosed