SCHEMBL10488583

SCHEMBL10488583

Cc1[nH]nc(N2CCN(Cc3ccccc3)CC2)c1C(=O)O

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 4/20 0.53
ALDH1A1 P00352 3/20 0.53
SMN1; SMN2 Q16637 2/20 0.53
KDM4E B2RXH2 3/20 0.51
MAPT P10636 2/20 0.51
MEN1 O00255 1/20 0.51
KMT2A Q03164 1/20 0.51
SMO Q99835 1/20 0.49
TSHR P16473 2/20 0.47
HTT P42858 1/20 0.47
HPGD P15428 1/20 0.47
DRD4 P21917 2/20 0.47
POLB P06746 1/20 0.47
HTR7 P34969 2/20 0.46
DRD2 P14416 1/20 0.46
DRD3 P35462 1/20 0.46
SIGMAR1 Q99720 1/20 0.46
GAA P10253 1/20 0.46
USP2 O75604 1/20 0.46
TP53 P04637 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10488589 0.87 SMN1; SMN2 (0.55) LMNAALDH1A1SMN1; SMN2KDM4EMAPT
SCHEMBL10488467 0.84 TTR (0.50) LMNAALDH1A1SMN1; SMN2KDM4EMAPT
SCHEMBL20438319 0.79 MEN1 (0.55) LMNAALDH1A1KDM4EMAPTMEN1
SCHEMBL10488580 0.77 HTT (0.50) ALDH1A1MAPTHTTHPGD
SCHEMBL10488632 0.76 HTT (0.53) ALDH1A1SMN1; SMN2KDM4EMAPTHTT
SCHEMBL10488586 0.74 LRRK2 (0.47) LMNAALDH1A1KDM4EMAPTMEN1
SCHEMBL13720391 0.72 ALDH1A1 (0.60) LMNAALDH1A1SMN1; SMN2KDM4EMAPT
SCHEMBL9778508 0.71 ALDH1A1 (0.59) LMNAALDH1A1SMN1; SMN2KDM4EMAPT
SCHEMBL7235226 0.71 HTR3E (0.61) LMNAALDH1A1SMN1; SMN2KDM4EMAPT
SCHEMBL27911478 0.71 ALDH1A1 (0.47) LMNAALDH1A1KDM4EDRD4POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4871737-A 3-Amino-5-methyl-1H-pyrazole-4-carboxylic acids and esters thereof as anticonvulsants muscle relaxants and anxiolytics A. H. ROBINS COMPANY, INCORPORATED (US) 1989-10-03 US disclosed
US-4826866-A 3-amino-5-methyl-1H-pyrazole-4-carboxylic acids and esters thereof as anticonvulsants, muscle relaxants and anxiolytics A. H. ROBINS COMPANY, INCORPORATED (US) 1989-05-02 US disclosed