SCHEMBL1049347

SCHEMBL1049347

CCCCCCCc1ccc(-c2ccc(CCCCCCC)cn2)nc1

nearest known ligand 0.71

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 9/20 0.71
SMN1; SMN2 Q16637 8/20 0.71
NPC1 O15118 7/20 0.71
MAPT P10636 5/20 0.71
STAT3 P40763 1/20 0.71
ATM Q13315 1/20 0.71
L3MBTL1 Q9Y468 4/20 0.64
CASP3 P42574 2/20 0.64
SENP8 Q96LD8 2/20 0.64
SENP7 Q9BQF6 2/20 0.64
SENP6 Q9GZR1 2/20 0.64
NFKB1 P19838 5/20 0.60
NFKB2 Q00653 4/20 0.60
RELA Q04206 4/20 0.60
MAPK1 P28482 2/20 0.60
TP53 P04637 2/20 0.54
POLB P06746 1/20 0.54
KDM4E B2RXH2 5/20 0.54
ALDH1A1 P00352 5/20 0.54
HPGD P15428 3/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1046569 1.00 RAB9A (0.71) RAB9ASMN1; SMN2NPC1MAPTSTAT3
SCHEMBL9081648 0.98 RAB9A (0.69) RAB9ASMN1; SMN2NPC1MAPTSTAT3
SCHEMBL9082721 0.94 RAB9A (0.65) RAB9ASMN1; SMN2NPC1MAPTSTAT3
SCHEMBL9083207 0.90 RAB9A (0.60) RAB9ASMN1; SMN2NPC1MAPTSTAT3
SCHEMBL10557531 0.89 RAB9A (0.82) RAB9ASMN1; SMN2NPC1MAPTSTAT3
SCHEMBL10558311 0.89 RAB9A (0.82) RAB9ASMN1; SMN2NPC1MAPTSTAT3
SCHEMBL10560635 0.89 RAB9A (0.82) RAB9ASMN1; SMN2NPC1MAPTSTAT3
SCHEMBL12622285 0.89 RAB9A (0.63) RAB9ASMN1; SMN2NPC1MAPTSTAT3
SCHEMBL10556991 0.89 RAB9A (0.82) RAB9ASMN1; SMN2NPC1MAPTSTAT3
SCHEMBL10555730 0.89 RAB9A (0.82) RAB9ASMN1; SMN2NPC1MAPTSTAT3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20170044392-A1 POLYMER COATING COMPRISING 2-METHOXYETHYL ACRYLATE UNITS SYNTHESIZED BY SURFACE-INITIATED ATOM TRANSFER RADICAL POLYMERIZATION UNIV DENMARK TECH DTU (DK) 2017-02-16 US disclosed
US-9346971-B2 Polymer coating comprising 2-methoxyethyl acrylate units synthesized by surface-initiated atom transfer radical polymerization TECHNICAL UNIVERSITY OF DENMARK (DK) 2016-05-24 US disclosed
EP-2453942-B1 POLYMER COATING COMPRISING 2-METHOXYETHYL ACRYLATE UNITS SYNTHESIZED BY SURFACE-INITIATED ATOM TRANSFER RADICAL POLYMERIZATION UNIV DENMARK TECH DTU (DK) 2014-08-13 EP disclosed
US-20120199825-A1 ORGANIC ELECTROLUMINESCENT DEVICE SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 2012-08-09 US disclosed
US-20120184029-A1 POLYMER COATING COMPRISING 2- METHOXYETHYL ACRYLATE UNITS SYNTHESIZED BY SURFACE-INITIATED ATOM TRANSFER RADICAL POLYMERIZATION TECHNICAL UNIVERSITY OF DENMARK (DK) 2012-07-19 US disclosed
EP-2453942-A2 POLYMER COATING COMPRISING 2-METHOXYETHYL ACRYLATE UNITS SYNTHESIZED BY SURFACE-INITIATED ATOM TRANSFER RADICAL POLYMERIZATION Technical University of Denmark (DK) 2012-05-23 EP disclosed
WO-2011006507-A2 POLYMER COATING COMPRISING 2-METHOXYETHYL ACRYLATE UNITS SYNTHESIZED BY SURFACE-INITIATED ATOM TRANSFER RADICAL POLYMERIZATION TECHNICAL UNIVERSITY OF DENMARK (DK) 2011-01-20 WO disclosed