SCHEMBL10499072

SCHEMBL10499072

NCCNC(=O)C1CCCOC1

nearest known ligand 0.44

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 4/20 0.44
DRD4 P21917 4/20 0.44
DRD2 P14416 3/20 0.44
HDAC3 O15379 1/20 0.40
HDAC1 Q13547 1/20 0.40
HDAC2 Q92769 1/20 0.40
ITGB3 P05106 5/20 0.39
ITGA2B P08514 5/20 0.39
NAAA Q02083 1/20 0.38
EPHX1 P07099 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.35
HSD17B10 Q99714 1/20 0.35
ALDH1A1 P00352 1/20 0.35
KEAP1 Q14145 1/20 0.34
NFE2L2 Q16236 1/20 0.34
GNAI3 P08754 1/20 0.34
GNAO1 P09471 1/20 0.34
GNAI1 P63096 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22170892 0.88 NAAA (0.48) HTR1ADRD4DRD2ITGB3ITGA2B
SCHEMBL16768104 0.85 HTR1A (0.45) HTR1ADRD4DRD2HDAC3HDAC1
SCHEMBL4679015 0.80 NAAA (0.50) ITGB3ITGA2BNAAAEPHX1SMN1; SMN2
SCHEMBL4678443 0.80 NAAA (0.55) ITGB3ITGA2BNAAAEPHX1SMN1; SMN2
SCHEMBL9558337 0.79 HTR1A (0.42) HTR1ADRD4DRD2NAAAALDH1A1
SCHEMBL10304069 0.78 NAAA (0.68) NAAAEPHX1GNAI3GNAO1GNAI1
SCHEMBL23419143 0.78 NAAA (0.58) ITGB3ITGA2BNAAAEPHX1SMN1; SMN2
SCHEMBL61158 0.78 NAAA (0.58) ITGB3ITGA2BNAAAEPHX1SMN1; SMN2
SCHEMBL19550760 0.77 HDAC3 (0.45) HTR1ADRD4DRD2HDAC3HDAC1
SCHEMBL19551083 0.77 HDAC3 (0.45) HTR1ADRD4DRD2HDAC3HDAC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0105838-B1 3-AMINOPROPOXYPHENYL DERIVATIVES, THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM Louis, William John (AU) 1989-06-21 EP disclosed
US-4661513-A 3-aminopropoxyphenyl derivatives, their preparation and pharmaceutical compositions containing them Louis, William John (AU) 1987-04-28 US disclosed
EP-0105838-A1 3-Aminopropoxyphenyl derivatives, their preparation and pharmaceutical compositions containing them Louis, William John (AU) 1984-04-18 EP disclosed