SCHEMBL10503100

SCHEMBL10503100

CCCCC1COC(c2ccc(C#N)cc2F)OC1

nearest known ligand 0.37

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CYP11B2 P19099 4/20 0.37
CYP19A1 P11511 2/20 0.36
CYP11B1 P15538 2/20 0.36
CYP17A1 P05093 1/20 0.36
HRH1 P35367 1/20 0.36
KCNH2 Q12809 1/20 0.36
DRD2 P14416 5/20 0.35
DRD3 P35462 5/20 0.35
GRM2 Q14416 2/20 0.35
SLC6A4 P31645 4/20 0.34
PSEN1 P49768 1/20 0.32
PSEN2 P49810 1/20 0.32
APH1B Q8WW43 1/20 0.32
NCSTN Q92542 1/20 0.32
APH1A Q96BI3 1/20 0.32
PSENEN Q9NZ42 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10501754 0.96 GRM2 (0.39) CYP11B2CYP19A1CYP11B1CYP17A1HRH1
SCHEMBL10502006 0.95 GRM2 (0.40) CYP11B2CYP19A1CYP11B1CYP17A1HRH1
SCHEMBL10779789 0.95 GRM2 (0.40) CYP11B2CYP19A1CYP11B1CYP17A1HRH1
SCHEMBL10776516 0.95 GRM2 (0.40) CYP11B2CYP19A1CYP11B1CYP17A1HRH1
SCHEMBL10501454 0.95 GRM2 (0.40) CYP11B2CYP19A1CYP11B1CYP17A1HRH1
SCHEMBL10502050 0.92 CYP11B2 (0.38) CYP11B2CYP19A1CYP11B1CYP17A1HRH1
SCHEMBL10501106 0.87 CYP11B2 (0.39) CYP11B2CYP19A1CYP11B1CYP17A1HRH1
SCHEMBL10502774 0.82 CYP11B2 (0.36) CYP11B2CYP19A1CYP11B1CYP17A1HRH1
SCHEMBL10779776 0.82 MGLL (0.40) CYP11B2CYP11B1
SCHEMBL10502495 0.81 CYP11B2 (0.35) CYP11B2CYP19A1CYP11B1CYP17A1HRH1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0154840-B1 LIQUID CRYSTAL COMPOUNDS MERCK PATENT GmbH (DE) 1989-01-25 EP disclosed
US-4704227-A DERIVATIVES OF 1,3-DIOXANE MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1987-11-03 US disclosed
EP-0154840-A2 Liquid crystal compounds MERCK PATENT GmbH (DE) 1985-09-18 EP disclosed