SCHEMBL10508364

SCHEMBL10508364

CCC(C)OC(=O)C(C(=O)O)c1csc(NC(=O)OC(C)(C)C)n1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ABCB1 P08183 1/20 0.40
PI4KB Q9UBF8 1/20 0.38
CA1 P00915 1/20 0.37
CA2 P00918 1/20 0.37
SMN1; SMN2 Q16637 2/20 0.37
CCR2 P41597 2/20 0.37
PTPRB P23467 1/20 0.36
LMNA P02545 1/20 0.36
KCNH2 Q12809 1/20 0.36
SIRT1 Q96EB6 1/20 0.35
SYK P43405 1/20 0.35
HDAC3 O15379 2/20 0.35
HDAC1 Q13547 2/20 0.35
HDAC2 Q92769 2/20 0.35
HDAC10 Q969S8 2/20 0.35
HDAC8 Q9BY41 2/20 0.35
ALDH1A1 P00352 2/20 0.34
MEN1 O00255 1/20 0.34
POLB P06746 1/20 0.34
MIF P14174 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10505216 0.83 CYP1A2 (0.39) CA1CA2SMN1; SMN2LMNAALDH1A1
SCHEMBL10505480 0.82 SMN1; SMN2 (0.50) SMN1; SMN2LMNAMEN1KMT2AMAPK1
SCHEMBL4899037 0.81 CCR2 (0.44) ABCB1PI4KBCA1CA2SMN1; SMN2
SCHEMBL10508353 0.81 SMN1; SMN2 (0.47) ABCB1PI4KBCA1CA2SMN1; SMN2
SCHEMBL10504410 0.80 SMN1; SMN2 (0.36) CA1CA2SMN1; SMN2CCR2LMNA
SCHEMBL10506393 0.78 MAPT (0.39) SMN1; SMN2LMNAALDH1A1POLB
SCHEMBL28334812 0.77 PI4KB (0.42) PI4KBCA1CA2CCR2PTPRB
SCHEMBL16748763 0.76 PI4KB (0.44) ABCB1PI4KBCA1CA2CCR2
SCHEMBL11186219 0.76 PI4KB (0.37) ABCB1PI4KBCA1CA2SMN1; SMN2
SCHEMBL11204633 0.76 PI4KB (0.42) PI4KBCA1CA2CCR2PTPRB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0168025-B1 PROCESS FOR PRODUCING AMINOTHIAZOLYLPROPENDICARBOXYLIC ACID MONOESTERS SHIONOGI & CO., LTD. (JP) 1989-09-27 EP disclosed
US-4652652-A PENICILLIN OR CEPHALOSPORIN INTERMEDIATE SHIONOGI & CO., LTD. (JP) 1987-03-24 US disclosed
EP-0168025-A1 Process for producing aminothiazolylpropendicarboxylic acid monoesters SHIONOGI & CO., LTD. (JP) 1986-01-15 EP disclosed