SCHEMBL10509705

SCHEMBL10509705

NC(=O)CN1C[C@H]2CCC[C@H]2C1=O

nearest known ligand 0.44

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
APEX1 P27695 1/20 0.44
BLM P54132 1/20 0.44
TSHR P16473 2/20 0.42
HTT P42858 1/20 0.41
FKBP1A P62942 1/20 0.37
RAB9A P51151 1/20 0.35
TP53 P04637 1/20 0.34
PER2 O15055 2/20 0.33
ACE P12821 2/20 0.32
DPP7 Q9UHL4 1/20 0.31
OPRM1 P35372 1/20 0.31
OPRL1 P41146 1/20 0.31
CYP2C19 P33261 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10509699 1.00 APEX1 (0.44) APEX1BLMTSHRHTTFKBP1A
SCHEMBL10509709 1.00 APEX1 (0.44) APEX1BLMTSHRHTTFKBP1A
SCHEMBL10509267 0.97 HTT (0.44) APEX1BLMTSHRHTTFKBP1A
SCHEMBL10509273 0.97 HTT (0.44) APEX1BLMTSHRHTTFKBP1A
SCHEMBL10510655 0.97 HTT (0.44) APEX1BLMTSHRHTTFKBP1A
SCHEMBL10510658 0.97 HTT (0.44) APEX1BLMTSHRHTTFKBP1A
SCHEMBL10509270 0.97 HTT (0.44) APEX1BLMTSHRHTTFKBP1A
SCHEMBL10764907 0.95 HTT (0.43) APEX1BLMTSHRHTTFKBP1A
SCHEMBL10508253 0.95 HTT (0.43) APEX1BLMTSHRHTTFKBP1A
SCHEMBL30876267 0.81 APEX1 (0.47) APEX1BLMTSHRHTTFKBP1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0213506-B1 Saturated cycloalkyl[c]pyrrole-2(1H)-acetic acid amides and derivatives thereof WARNER-LAMBERT COMPANY (US) 1989-02-15 EP claimed
EP-0213506-A1 Saturated cycloalkyl[c]pyrrole-2(1H)-acetic acid amides and derivatives thereof WARNER-LAMBERT COMPANY (US) 1987-03-11 EP claimed
US-4621097-A COGNITION ACTIVATORS WARNER-LAMBERT COMPANY (US) 1986-11-04 US claimed
EP-0213506-B1 Saturated cycloalkyl[c]pyrrole-2(1H)-acetic acid amides and derivatives thereof WARNER-LAMBERT COMPANY (US) 1989-02-15 EP disclosed
EP-0213506-A1 Saturated cycloalkyl[c]pyrrole-2(1H)-acetic acid amides and derivatives thereof WARNER-LAMBERT COMPANY (US) 1987-03-11 EP disclosed
US-4621097-A COGNITION ACTIVATORS WARNER-LAMBERT COMPANY (US) 1986-11-04 US disclosed