SCHEMBL10510799

SCHEMBL10510799

O=C(OCCN1CCCCC1)c1ccccc1Nc1ccnc2cc(C(F)(F)F)ccc12

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RXFP1 Q9HBX9 1/20 0.49
SLC6A2 P23975 2/20 0.48
PDE4D Q08499 2/20 0.48
KCNH2 Q12809 2/20 0.48
HTR2A P28223 1/20 0.48
OPRK1 P41145 1/20 0.48
HTR2B P41595 1/20 0.48
SLC6A3 Q01959 1/20 0.48
CYP1A2 P05177 3/20 0.47
CYP2C9 P11712 3/20 0.47
CYP3A4 P08684 2/20 0.47
MAPK1 P28482 2/20 0.47
HSD17B10 Q99714 2/20 0.47
HPGD P15428 2/20 0.47
CYP2C19 P33261 2/20 0.47
ALDH1A1 P00352 2/20 0.47
CYP2D6 P10635 2/20 0.47
KDM4E B2RXH2 1/20 0.47
MLNR O43193 1/20 0.47
ABCB11 O95342 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10631435 1.00 RXFP1 (0.49) RXFP1SLC6A2PDE4DKCNH2HTR2A
Florifenine SCHEMBL29400044 0.99 SLC6A2 (0.49) RXFP1SLC6A2PDE4DKCNH2HTR2A
Florifenine SCHEMBL379372 0.99 SLC6A2 (0.49) RXFP1SLC6A2PDE4DKCNH2HTR2A
SCHEMBL10626075 0.95 CYP1A2 (0.48) RXFP1SLC6A2PDE4DKCNH2HTR2A
SCHEMBL10510019 0.95 CYP1A2 (0.48) RXFP1SLC6A2PDE4DKCNH2HTR2A
SCHEMBL10509149 0.94 CYP1A2 (0.49) RXFP1SLC6A2PDE4DKCNH2HTR2A
Antrafenine SCHEMBL29623495 0.89 HTR4 (0.51) SLC6A2PDE4DKCNH2HTR2AOPRK1
Antrafenine SCHEMBL24297 0.89 HTR4 (0.51) SLC6A2PDE4DKCNH2HTR2AOPRK1
SCHEMBL10510990 0.87 CYP3A4 (0.48) SLC6A2PDE4DKCNH2CYP1A2CYP2C9
SCHEMBL10509334 0.87 CYP3A4 (0.63) SLC6A2PDE4DKCNH2CYP1A2CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0094065-B1 2-AMINOBENZOIC ACID DERIVATIVES, A PROCESS FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS FERRER INTERNACIONAL, S.A. (ES) 1989-12-20 EP disclosed
US-4767767-A ANALGESIC, ANTIINFLAMMATORY AGENT FERRER INTERNACIONAL S.A. (ES) 1988-08-30 US disclosed
EP-0094065-A2 2-Aminobenzoic acid derivatives, a process for their preparation and pharmaceutical compositions FERRER INTERNACIONAL, S.A. (ES) 1983-11-16 EP disclosed