SCHEMBL10512751

SCHEMBL10512751

CCCCCc1ccc(-c2ccc(C#Cc3ccc(CC)cc3)c(F)c2F)cc1.CCCCc1ccc(-c2ccc(C#Cc3ccc(CC)cc3)c(F)c2F)cc1.CCCc1ccc(-c2ccc(C#Cc3ccc(CC)cc3)c(F)c2F)cc1.CCc1ccc(C#Cc2ccc(-c3ccc(C)cc3)c(F)c2F)cc1.CCc1ccc(C#Cc2ccc(-c3ccc(CC)cc3)c(F)c2F)cc1

nearest known ligand 0.40

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.40
HSD17B10 Q99714 1/20 0.40
RARB P10826 4/20 0.38
NPC1 O15118 1/20 0.35
RAB9A P51151 1/20 0.35
ATM Q13315 1/20 0.35
HSD11B1 P28845 4/20 0.35
MPL P40238 5/20 0.35
FFAR1 O14842 3/20 0.34
FAAH O00519 1/20 0.33
RARA P10276 1/20 0.33
RARG P13631 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10519630 1.00 TSHR (0.40) TSHRHSD17B10RARBNPC1RAB9A
SCHEMBL10511580 1.00 TSHR (0.40) TSHRHSD17B10RARBNPC1RAB9A
SCHEMBL10511143 1.00 TSHR (0.40) TSHRHSD17B10RARBNPC1RAB9A
SCHEMBL9508912 0.93 TSHR (0.45) TSHRHSD17B10RARBNPC1RAB9A
SCHEMBL9512364 0.93 TSHR (0.45) TSHRHSD17B10RARBNPC1RAB9A
SCHEMBL9508830 0.92 HSD17B10 (0.46) TSHRHSD17B10RARBHSD11B1MPL
SCHEMBL9512324 0.92 FFAR1 (0.40) TSHRHSD17B10RARBNPC1RAB9A
SCHEMBL9512306 0.92 HSD17B10 (0.46) TSHRHSD17B10RARBHSD11B1MPL
SCHEMBL9511284 0.92 FFAR1 (0.40) TSHRHSD17B10RARBNPC1RAB9A
SCHEMBL9510180 0.91 TSHR (0.40) TSHRHSD17B10RARBHSD11B1MPL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0308438-A1 Liquid crystal phase containing tolanes. MERCK PATENT GMBH (DE) 1989-03-29 EP disclosed
WO-1988007514-A1 TOLANES MERCK Patent Gesellschaft mit beschränkter Haftung (DE) 1988-10-06 WO disclosed