SCHEMBL10518481

SCHEMBL10518481

CN1CCC(C(=O)C2c3cc(Cl)ccc3NC(=O)c3ccccc32)CC1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HRH4 Q9H3N8 2/20 0.40
HRH3 Q9Y5N1 2/20 0.40
ATM Q13315 1/20 0.40
CHEK1 O14757 1/20 0.40
MAPT P10636 3/20 0.39
CYP1A2 P05177 2/20 0.39
CYP2C9 P11712 2/20 0.39
TSHR P16473 2/20 0.39
CYP2C19 P33261 2/20 0.39
TP53 P04637 1/20 0.39
ALOX15 P16050 1/20 0.39
CASP1 P29466 1/20 0.39
RECQL P46063 1/20 0.39
SLC8B1 Q6J4K2 1/20 0.39
MEN1 O00255 3/20 0.37
KMT2A Q03164 3/20 0.37
IDO1 P14902 1/20 0.37
TDO2 P48775 1/20 0.37
TGM2 P21980 1/20 0.37
DRD4 P21917 2/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10483573 0.88 MEN1 (0.40) MAPTCYP1A2MEN1KMT2AIDO1
SCHEMBL10516167 0.83 PARP1 (0.37) MAPTCYP1A2TSHRCASP1MEN1
SCHEMBL10516856 0.82 CSNK1G1 (0.41) MAPTCASP1DRD4LMNAHSD17B10
SCHEMBL10515295 0.80 PARP1 (0.39) MAPTCYP1A2TSHRCASP1MEN1
SCHEMBL10515664 0.79 POLB (0.38) CYP1A2CYP2C9TSHRCYP2C19CASP1
SCHEMBL10514837 0.78 ALDH1A1 (0.38) MEN1KMT2A
SCHEMBL10517669 0.78 DAO (0.38) MAPTMEN1KMT2ADRD4LMNA
SCHEMBL10514845 0.76 CHRM2 (0.40) MAPTCASP1CHRM2CHRM4CYP3A4
SCHEMBL10515428 0.76 ALDH1A1 (0.39) HRH3MAPTMEN1KMT2AIDO1
SCHEMBL10516012 0.76 POLB (0.37) CYP1A2CYP2C9TSHRCYP2C19CASP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0326526-A1 Aminoketones of substituted dibenzo- and pyridobenzo-azepinones and pharmaceutical compositions ISTITUTO DE ANGELI S.p.A. (IT) 1989-08-02 EP disclosed