SCHEMBL10521682

SCHEMBL10521682

O=C(O)C(CCCCCCc1ccccc1)Cc1cccc2ccccc12

nearest known ligand 0.60

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 1/20 0.51
PTGES O14684 1/20 0.51
ALOX5 P09917 1/20 0.51
PPARG P37231 1/20 0.51
HRH4 Q9H3N8 1/20 0.49
FOLH1 Q04609 3/20 0.49
KMT2A Q03164 1/20 0.49
CTNNB1 P35222 1/20 0.48
GRIK1 P39086 1/20 0.47
METAP2 P50579 1/20 0.45
CPB2 Q96IY4 1/20 0.44
TDP1 Q9NUW8 1/20 0.44
BID P55957 1/20 0.44
BCL2L1 Q07817 1/20 0.44
MCL1 Q07820 1/20 0.44
BAK1 Q16611 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10521472 0.99 SIGMAR1 (0.52) SIGMAR1PTGESALOX5PPARGHRH4
SCHEMBL10521941 0.95 SIGMAR1 (0.53) SIGMAR1PTGESALOX5PPARGHRH4
SCHEMBL10522911 0.84 SIGMAR1 (0.49) SIGMAR1PTGESALOX5PPARGHRH4
SCHEMBL7280252 0.83 CTNNB1 (0.52) HRH4FOLH1KMT2ACTNNB1TDP1
SCHEMBL7280245 0.83 CTNNB1 (0.52) HRH4FOLH1KMT2ACTNNB1TDP1
SCHEMBL5953914 0.82 FOLH1 (0.66) HRH4FOLH1CTNNB1TDP1
SCHEMBL1858161 0.82 KMT2A (0.52) SIGMAR1HRH4KMT2ACTNNB1GRIK1
SCHEMBL10522072 0.82 HRH4 (0.50) SIGMAR1PTGESALOX5PPARGHRH4
SCHEMBL7352579 0.82 CYP1A2 (0.65) PPARGHRH4FOLH1KMT2ACTNNB1
SCHEMBL10521559 0.81 FOLH1 (0.68) PTGESALOX5PPARGFOLH1GRIK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4863904-A Dipeptides as renin inhibitors KISSEI PHARMACEUTICAL CO., LTD. (JP) 1989-09-05 US disclosed
EP-0181110-A2 Histidine derivatives as renin inhibitors Kissei Pharmaceutical Co. Ltd. (JP) 1986-05-14 EP disclosed